Cover Image

Synthesis and Biological Evaluation of Novel Cationic Rhenium and Technetium-99m Complexes Bearing Quinazoline Derivative for Epidermal Growth Factor Receptor Targeting

<b>Background/Objectives:</b> Epidermal growth factor receptor (EGFR) plays a vital role in cell proliferation and survival, with its overexpression linked to various malignancies, including non-small cell lung cancer (NSCLC). Although EGFR tyrosine kinase inhibitors (TKIs) are a key the...

Full description

Saved in:

Bibliographic Details
Main Authors:	Sotiria Triantopoulou (Author), Ioanna Roupa (Author), Antonio Shegani (Author), Nektarios N. Pirmettis (Author), Georgia I. Terzoudi (Author), Aristeidis Chiotellis (Author), Maria Tolia (Author), John Damilakis (Author), Ioannis Pirmettis (Author), Maria Paravatou-Petsota (Author)
Format:	Book
Published:	MDPI AG, 2024-09-01T00:00:00Z.
Subjects:	article
Online Access:	Connect to this object online.
Tags:	Add Tag No Tags, Be the first to tag this record!

Similar Items

Synthesis and Evaluation of <sup>99m</sup>Tc(CO)<sub>3</sub> Complexes with Ciprofloxacin Dithiocarbamate for Infection Imaging
by: Afroditi Papasavva, et al.
Published: (2024)

Radiolabeling of cidofovir with technetium-99m and biodistribution studies
by: Raquel Gregorio Arribada, et al.
Published: (2020)

The purity identification and radiolabeling of α-mangostin with technetium-99m
by: Muchtaridi Muchtaridi, et al.
Published: (2020)

Technetium-99m-labeled genistein as a potential radical scavenging agent
by: Danni Ramdhani, et al.
Published: (2019)

Labelling of human serum albumin (HSA)-nanospheres with technetium-99m radionuclide
by: Nanny Kartini Oekar, et al.
Published: (2008)

Technetium Tc 99m tilmanocept fails to detect sentinel lymph nodes in endometrial cancer
by: Ravali A. Reddy, et al.
Published: (2022)

A new two-strip TLC method for the quality control of technetium-99m mercaptoacetyl-triglycine (99mTc-MAG3)
by: Marietta Straub, et al.
Published: (2018)

The optimization method for synthesis of technetium-99m-luteolin as radiotracer in the development of cancer drugs from flavonoid
by: Danni Ramdhani, et al.
Published: (2020)

99m Technetium-HMPAO-labeled platelet scan in practice: Preparation, quality control, and biodistribution studies
by: Mahdieh Parvizi, et al.
Published: (2022)

Brain targeting efficiency of intranasal clozapine-loaded mixed micelles following radio labeling with Technetium-99m
by: Sinar Sayed, et al.
Published: (2021)

Cholecystokinin-2 Receptor Targeting with Novel C-terminally Stabilized HYNIC-Minigastrin Analogs Radiolabeled with Technetium-99m
by: Maximilian Klingler, et al.
Published: (2019)

Fusion-Based Neutron Generator Production of Tc-99m and Tc-101: A Prospective Avenue to Technetium Theranostics
by: Edward J. Mausolf, et al.
Published: (2021)

Computer-Aided Drug Design and Synthesis of Rhenium Clotrimazole Antimicrobial Agents
by: Youri Cortat, et al.
Published: (2023)

Cutaneous squamous cell carcinoma of the lip successfully treated with Rhenium-188 brachytherapy
by: Chiara Sabbadini, et al.
Published: (2023)

Technetium-99m sestamibi retention in skeletal muscles, a potential indicator of mitochondrial function and anaerobic threshold in patients with type 2 diabetes
by: Shinji Sato, et al.
Published: (2015)

Residence Time Distribution (RTD) model of water flooding in vertical sand column using Technetium-99m as the radiotracer / Noraishah Othman ... [et al.]
by: Othman, Noraishah, et al.
Published: (2022)

Double serum sampled glomerular filtration rate measurement with technetium-99m diethylenetriamine-penta acetate for evaluation of renal functions in patients with psoriasis vulgaris
by: Rukiye Yasak Guner, et al.
Published: (2021)

Injeção intraoperatória de dextran-500-99m_tecnécio para identificação do linfonodo sentinela em câncer de mama Intraoperative injection of technetium-99m-dextran 500 for the identification of sentinel lymph node in breast cancer
by: Gerson Jacob Delazeri, et al.
Published: (2010)

Bowel excretion of Technetium-99mL, L-Ethylene dicysteine masquerading as a dilated ureter in a case of pelvi-ureteric junction obstruction: Case report and review
by: Prabudh Goel, et al.
Published: (2019)

Antimicrobial Activity of Rhenium Di- and Tricarbonyl Diimine Complexes: Insights on Membrane-Bound <i>S. aureus</i> Protein Binding
by: Kevin Schindler, et al.
Published: (2022)

Inhibition of the Hepatic Uptake of <sup>99m</sup>Tc-Tetrofosmin Using an Organic Cation Transporter Blocker
by: Kodai Nishi, et al.
Published: (2021)

Quinazolinone and Quinazoline Derivatives
Published: (2020)

Avaliação da densidade mamográfica e da captação cintimamográfica de sestamibi-99mTecnécio, em mulheres na pós-menopausa sob terapia hormonal Evaluation of mammographic density and of scinti-mammographic uptake of sestamibi-99mTechnetium in postmenopausal women under hormonal treatment
by: Jorge Nahás Neto
Published: (2004)

TrisOxine abiotic siderophores for technetium complexation: radiolabeling and biodistribution studies
by: Julien Leenhardt, et al.
Published: (2023)

Quinazoline pharmacophore in therapeutic medicine
by: Olayinka Oyewale Ajani, et al.
Published: (2016)

Correction: Klingler, M., et al. Cholecystokinin-2 Receptor Targeting with Novel C-terminally Stabilized HYNIC-Minigastrin Analogs Radiolabeled with Technetium-99m. <i>Pharmaceuticals</i> 2019, <i>12</i>, 13
by: Maximilian Klingler, et al.
Published: (2019)

Assessment of exposure of workers to ionizing radiation from radioiodine and technetium in nuclear medicine departmental facilities
by: Grażyna Krajewska, et al.
Published: (2013)

Synthesis and anticancer activity of new quinazoline derivatives
by: Hatem A. Abuelizz, et al.
Published: (2017)

VEGFR-2 inhibitors and apoptosis inducers: synthesis and molecular design of new benzo[g]quinazolin bearing benzenesulfonamide moiety
by: Mostafa M. Ghorab, et al.
Published: (2017)

Deciphering the enzymatic target of a new family of antischistosomal agents bearing a quinazoline scaffold using complementary computational tools
by: Victor Sebastian-Perez, et al.
Published: (2020)

Design, Synthesis, Pharmacological Evaluation of Quinazolin-4(3H)-Ones Bearing Urea Functionality as Potential VEGFR-2 Inhibitors
by: Al-Sanea MM, et al.
Published: (2024)

Synthesis of chalcone incorporated quinazoline derivatives as anticancer agents
by: Sapavat Madhavi, et al.
Published: (2017)

Design and Molecular Docking Studies of Quinazoline Derivatives as Antiproliferation
by: Anita Puspa Widiyana, et al.
Published: (2018)

Magnesium-Molybate Compounds as Matrix for 99Mo/99mTc Generators
by: Fabiola Monroy-Guzman, et al.
Published: (2011)

Introduction of pyrrolidineoxy or piperidineamino group at the 4-position of quinazoline leading to novel quinazoline-based phosphoinositide 3-kinase delta (PI3Kδ) inhibitors
by: Minhang Xin, et al.
Published: (2018)

Quinazoline analogues as cytotoxic agents; QSAR, docking, and in silico studies
by: Leila Emami, et al.
Published: (2021)

Medicinal Chemistry of Quinazolines as Anticancer Agents Targeting Tyrosine Kinases
by: Mohamed F. Zayed
Published: (2023)

Potential Positive Effects of COVID-19 on Cancer Care: A Window of Opportunity
by: Emmanouil Damilakis
Published: (2022)

A Novel Therapeutic Strategy for Cancer Using Phosphatidylserine Targeting Stearylamine-Bearing Cationic Liposomes
by: Manjarika De, et al.
Published: (2018)

Novel Thiazole-Fused [4,5-<i>g</i>] or [5,4-<i>g</i>]Quinazolin-8-ones and Their Quinazoline Analogues: Synthesis and Biological Evaluation
by: Nathan Broudic, et al.
Published: (2024)