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Computationally driven discovery of phenyl(piperazin-1-yl)methanone derivatives as reversible monoacylglycerol lipase (MAGL) inhibitors

Monoacylglycerol lipase (MAGL) is an attractive therapeutic target for many pathologies, including neurodegenerative diseases, cancer as well as chronic pain and inflammatory pathologies. The identification of reversible MAGL inhibitors, devoid of the side effects associated to prolonged MAGL inacti...

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Bibliographic Details
Main Authors:	Giulio Poli (Author), Margherita Lapillo (Author), Vibhu Jha (Author), Nayla Mouawad (Author), Isabella Caligiuri (Author), Marco Macchia (Author), Filippo Minutolo (Author), Flavio Rizzolio (Author), Tiziano Tuccinardi (Author), Carlotta Granchi (Author)
Format:	Book
Published:	Taylor & Francis Group, 2019-01-01T00:00:00Z.
Subjects:	article
Online Access:	Connect to this object online.
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