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Exploring Kinase Inhibition Properties of 9<i>H</i>-pyrimido[5,4-<i>b</i>]- and [4,5-<i>b</i>]indol-4-amine Derivatives

We previously highlighted the interest in 6,5,6-fused tricyclic analogues of 4-aminoquinazolines as kinase inhibitors in the micromolar to the nanomolar range of IC<sub>50</sub> values. For the generation of chemical libraries, the formamide-mediated cyclization of the cyanoamidine precu...

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Main Authors:	Yvonnick Loidreau (Author), Carole Dubouilh-Benard (Author), Marie-Renée Nourrisson (Author), Nadège Loaëc (Author), Laurent Meijer (Author), Thierry Besson (Author), Pascal Marchand (Author)
Format:	Book
Published:	MDPI AG, 2020-05-01T00:00:00Z.
Subjects:	article
Online Access:	Connect to this object online.
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