Transport Characteristics of Tryptanthrin and its Inhibitory Effect on P-gp and MRP2 in Caco-2 Cells
Purpose. Tryptanthrin, an indole quinazoline alkaloid with multiple medical activities, has been recently under preclinical development as an anti-tuberculosis and anti-tumor drug. The aims of this study are to characterize the intestinal transport of tryptanthrin in Caco-2 cells, to determine wheth...
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Main Authors: | Xingang Zhu (Author), Xuelian Zhang (Author), Guo Ma (Author), Junkai Yan (Author), Honghai Wang (Author), Qing Yang (Author) |
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Format: | Book |
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Frontiers Media S.A.,
2011-08-01T00:00:00Z.
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Online Access: | Connect to this object online. |
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