Development of Novel Fluorinated Polyphenols as Selective Inhibitors of DYRK1A/B Kinase for Treatment of Neuroinflammatory Diseases including Parkinson's Disease
Natural polyphenol derivatives such as those found in green tea have been known for a long time for their useful therapeutic activity. Starting from EGCG, we have discovered a new fluorinated polyphenol derivative (<b>1c</b>) characterized by improved inhibitory activity against DYRK1A/B...
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Main Authors: | Gian Luca Araldi (Author), Yu-Wen Hwang (Author) |
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Format: | Book |
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MDPI AG,
2023-03-01T00:00:00Z.
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Online Access: | Connect to this object online. |
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