Contribution of Active and Inactive States of the Human 5-HT4d Receptor to the Functional Activities of 5-HT4-Receptor Agonists
In the present study, binding affinities of 5-hydroxytryptamine-4 (5-HT4) ligands for the human 5-HT4d receptor were determined using the agonist [3H]5-HT and the selective 5-HT4 antagonist [3H]GR113,808. We also compared the affinity differences between [3H]5-HT binding (KH) and [3H]GR113,808 bindi...
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Main Authors: | Tadayoshi Mikami (Author), Hiromi Sugimoto (Author), Rie Naganeo (Author), Takashi Ohmi (Author), Toshiyuki Saito (Author), Hiroyuki Eda (Author) |
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Format: | Book |
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Elsevier,
2008-01-01T00:00:00Z.
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Online Access: | Connect to this object online. |
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