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Blocking the CGRP Receptor: Differences across Human Vascular Beds

Multiple drugs targeting the calcitonin gene-related peptide (CGRP) receptor have been developed for the treatment of migraine. Here, the effect of the small-molecule CGRP receptor antagonist zavegepant (0.1 nM-1 µM) on CGRP-induced relaxation in isolated human coronary arteries (HCAs) was investiga...

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Bibliographic Details
Main Authors:	Tessa de Vries (Author), Deirdre M. Boucherie (Author), Antoon van den Bogaerdt (Author), A. H. Jan Danser (Author), Antoinette MaassenVanDenBrink (Author)
Format:	Book
Published:	MDPI AG, 2023-07-01T00:00:00Z.
Subjects:	article
Online Access:	Connect to this object online.
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