Impact of drug distribution into adipose on tissue function: The cholesteryl ester transfer protein (CETP) inhibitor anacetrapib as a test case
Abstract Anacetrapib is an inhibitor of cholesteryl ester transfer protein (CETP) previously under development as a lipid‐modifying agent that reduces LDL‐cholesterol and increases HDL‐cholesterol in hypercholesterolemic patients. Anacetrapib demonstrates a long terminal half‐life and accumulates in...
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Main Authors: | Douglas G. Johns (Author), Sheng‐Ping Wang (Author), Raymond Rosa (Author), James Hubert (Author), Suoyu Xu (Author), Ying Chen (Author), Thomas Bateman (Author), Robert O. Blaustein (Author) |
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Format: | Book |
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Wiley,
2019-12-01T00:00:00Z.
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Online Access: | Connect to this object online. |
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