Design, synthesis, and anticonvulsant effects evaluation of nonimidazole histamine H3 receptor antagonists/inverse agonists containing triazole moiety
Histamine H3 receptors (H3R) antagonists/inverse agonists are becoming a promising therapeutic approach for epilepsy. In this article, novel nonimidazole H3R antagonists/inverse agonists have been designed and synthesised via hybriding the H3R pharmacophore (aliphatic amine with propyloxy chain) wit...
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Main Authors: | Mingxia Song (Author), Rui Yan (Author), Yanhui Zhang (Author), Dongfu Guo (Author), Naiming Zhou (Author), XianQing Deng (Author) |
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Format: | Book |
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Taylor & Francis Group,
2020-01-01T00:00:00Z.
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Online Access: | Connect to this object online. |
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