Synthesis and Bioactivity of Thiazolethioacetamides as Potential Metallo-β-Lactamase Inhibitors
Metallo-β-lactamase (MβLs) mediated antibiotic resistance seriously threatens the treatment of bacterial diseases. Recently, we found that thioacetamides can be a potential MβL inhibitor skeleton. In order to improve the information of the skeleton, twelve new thiazolethioacetamides were designed by...
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Main Authors: | Yi-Lin Zhang (Author), Yong Yan (Author), Xue-Jun Wang (Author), Ke-Wu Yang (Author) |
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Format: | Book |
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MDPI AG,
2020-02-01T00:00:00Z.
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