The Impact of the Secondary Binding Pocket on the Pharmacology of Class A GPCRs
G-protein coupled receptors (GPCRs) are considered important therapeutic targets due to their pathophysiological significance and pharmacological relevance. Class A receptors represent the largest group of GPCRs that gives the highest number of validated drug targets. Endogenous ligands bind to the...
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Main Authors: | Attila Egyed (Author), Dóra Judit Kiss (Author), György M. Keserű (Author) |
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Format: | Book |
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Frontiers Media S.A.,
2022-03-01T00:00:00Z.
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