Search Results - "Medicinal Chemistry"

New sulfonamides containing organometallic-acylhydrazones: synthesis, characterisation and biological evaluation as inhibitors of human carbonic anhydrases by Yosselin Huentupil, Luis Peña, Néstor Novoa, Emanuela Berrino, Rodrigo Arancibia, Claudiu T. Supuran

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Antifungal and anti-biofilm effects of hydrazone derivatives on Candida spp by Pierre Popczyk, Alina Ghinet, Clovis Bortolus, Laure Kamus, Marc F. Lensink, Jérôme de Ruyck, Boualem Sendid, Faustine Dubar

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Novel thiazolidinone-containing compounds, without the well-known sulphonamide zinc-binding group acting as human carbonic anhydrase IX inhibitors by Özlen Güzel-Akdemir, Andrea Angeli, Kübra Demir, Claudiu T. Supuran, Atilla Akdemir

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ALDEFLUOR activity, ALDH isoforms, and their clinical significance in cancers by Jiang-Jie Duan, Jiao Cai, Lei Gao, Shi-Cang Yu

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Application of Chiral Piperidine Scaffolds in Drug Design by Qiu-Shi Chen, Jian-Qi Li, Qing-Wei Zhang

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Synthesis of new pyridothienopyrimidinone and pyridothienotriazolopyrimidine derivatives as pim-1 inhibitors by Hala B. El-Nassan, Bassem H. Naguib, Engy A. Beshay

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Models of enzyme inhibition and apparent dissociation constants from kinetic analysis to study the differential inhibition of aldose reductase by Francesco Balestri, Mario Cappiello, Roberta Moschini, Umberto Mura, Antonella Del-Corso

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Improved in vitro potency of Clofazimine derivatives against Neisseria species by Masahide Yano, Jessica M. Lawson-Rulli, Reilly M. Coates, Jennifer Heldring, Marvin J. Miller, Rui Liu

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Naphthoquinone amino acid derivatives, synthesis and biological activity as proteasome inhibitors by Mauro Marastoni, Claudio Trapella, Alessandra Scotti, Anna Fantinati, Valeria Ferretti, Erika Marzola, Gallerani Eleonora, Riccardo Gavioli, Delia Preti

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Exosomes in head and neck cancer. Updating and revisiting by Samuel Rodríguez Zorrilla, Abel García García, Andrés Blanco Carrión, Pilar Gándara Vila, Manuel Somoza Martín, Mercedes Gallas Torreira, Mario Pérez Sayans

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Pyrimidine analogues for the management of neurodegenerative diseases by Swati Pant, Anandi Kapri, Sumitra Nain

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Development of a cheminformatics platform for selectivity analyses of carbonic anhydrase inhibitors by Giulio Poli, Salvatore Galati, Adriano Martinelli, Claudiu T. Supuran, Tiziano Tuccinardi

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Prospective mode of action of Ivermectin: SARS-CoV-2 by Vaishali M. Patil, Saroj Verma, Neeraj Masand

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An overview of carbohydrate-based carbonic anhydrase inhibitors by Doretta Cuffaro, Elisa Nuti, Armando Rossello

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Fluoroenesulphonamides: N-sulphonylurea isosteres showing nanomolar selective cancer-related transmembrane human carbonic anhydrase inhibition by Benoit Métayer, Andrea Angeli, Agnès Mingot, Kévin Jouvin, Gwilherm Evano, Claudiu T. Supuran, Sébastien Thibaudeau

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Echinocandins - structure, mechanism of action and use in antifungal therapy by Mateusz Szymański, Sandra Chmielewska, Urszula Czyżewska, Marta Malinowska, Adam Tylicki

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Identification of cisplatin-binding sites on the large cytoplasmic loop of the Na+/K+-ATPase by Jaroslava Šeflová, Petra Čechová, Tereza Štenclová, Marek Šebela, Martin Kubala

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An overview: metal-based inhibitors of urease by Wei Yang, Zhiyun Peng, Guangcheng Wang

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Research progress of natural products and their derivatives against Alzheimer's disease by Jin-Ying Liu, Hong-Yan Guo, Zhe-Shan Quan, Qing-Kun Shen, Hong Cui, Xiaoting Li

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Discovery of new acetylcholinesterase inhibitors for Alzheimer's disease: virtual screening and in vitro characterisation by Benoit David, Pascal Schneider, Philipp Schäfer, Jörg Pietruszka, Holger Gohlke

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