Search Results - "Medicinal Chemistry"

Targeting carbonic anhydrase IX and XII isoforms with small molecule inhibitors and monoclonal antibodies by Mateusz Kciuk, Adrianna Gielecińska, Somdutt Mujwar, Mariusz Mojzych, Beata Marciniak, Rafał Drozda, Renata Kontek

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5-(Sulfamoyl)thien-2-yl 1,3-oxazole inhibitors of carbonic anhydrase II with hydrophilic periphery by Stanislav Kalinin, Alexander Kovalenko, Annika Valtari, Alessio Nocentini, Maxim Gureev, Arto Urtti, Mikhail Korsakov, Claudiu T. Supuran, Mikhail Krasavin

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Diaryl ethers with carboxymethoxyphenacyl motif as potent HIV-1 reverse transcriptase inhibitors with improved solubility by Tomasz Frączek, Rafał Kamiński, Agnieszka Krakowiak, Evelien Naessens, Bruno Verhasselt, Piotr Paneth

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Toxicity evaluation of sulfamides and coumarins that efficiently inhibit human carbonic anhydrases by Ashok Aspatwar, Emanuela Berrino, Silvia Bua, Fabrizio Carta, Clemente Capasso, Seppo Parkkila, Claudiu T. Supuran

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Inhibitory activity against carbonic anhydrase IX and XII as a candidate selection criterion in the development of new anticancer agents by Mikhail Krasavin, Stanislav Kalinin, Tatiana Sharonova, Claudiu T. Supuran

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A Comprehensive Review on Chemical Synthesis and Chemotherapeutic Potential of 3-Heteroaryl Fluoroquinolone Hybrids by Halyna Hryhoriv, Sergiy M. Kovalenko, Marine Georgiyants, Lyudmila Sidorenko, Victoriya Georgiyants

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Taccalonolides: Structure, semi-synthesis, and biological activity by Yan Li, Yu-Feng Du, Feng Gao, Jin-Bu Xu, Ling-Li Zheng, Gang Liu, Yu Lei

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1-(Piperidin-3-yl)thymine amides as inhibitors of M. tuberculosis thymidylate kinase by Yanlin Jian, Martijn D. P. Risseeuw, Mathy Froeyen, Lijun Song, Davie Cappoen, Paul Cos, Hélène Munier-Lehmann, Serge van Calenbergh

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Bulge oligonucleotide as an inhibitory agent of bacterial topoisomerase I by Zhaoqi Yang, Tuoyu Jiang, Hanshi Zhong, Yu Kang

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Synthesis and structure-activity relationships for some novel diflapolin derivatives with benzimidazole subunit by Lisa Vieider, Eva Zoeller, Erik Romp, Martin Schoenthaler, Victor Hernández-Olmos, Veronika Temml, Thomas Hasenoehrl, Daniela Schuster, Oliver Werz, Ulrike Garscha, Barbara Matuszczak

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Recent Advance in the biological activity of synephrine in Citri Reticulatae Pericarpium by Yue-Chang Huang, Jia-Min Li, Bai-Zhong Chen, Xing-Min Zhang, Ri-Hui Wu, Pan-Pan Wu, Chen Li, Wen-Hua Chen

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Discovery and efficacy study of an ALK inhibitor AMX6001 in anaplastic large cell lymphoma Karpas299 mice models by Debasis Das, Lingzhi Xie, Dandan Qiao, Yuxi Cao, Jianhe Jia, Yong Li, Jian Hong

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The insulin-degrading enzyme as a link between insulin and neuropeptides metabolism by Dorota Wacławczyk, Jerzy Silberring, Giuseppe Grasso

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Synthetic Imidazopyridine-Based Derivatives as Potential Inhibitors against Multi-Drug Resistant Bacterial Infections: A Review by Bharat Kumar Reddy Sanapalli, Akram Ashames, Dilep Kumar Sigalapalli, Afzal B. Shaik, Richie R. Bhandare, Vidyasrilekha Yele

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Calendula in modern medicine: Advancements in wound healing and drug delivery applications by Ovinuchi Ejiohuo, Samson Folami, Abdulkadir Yusif Maigoro

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Crystal structure of the human carbonic anhydrase II adduct with 1-(4-sulfamoylphenyl-ethyl)-2,4,6-triphenylpyridinium perchlorate, a membrane-impermeant, isoform selective inhibit... by Vincenzo Alterio, Davide Esposito, Simona Maria Monti, Claudiu T. Supuran, Giuseppina De Simone

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The Structures and Binding Modes of Small-Molecule Inhibitors of <i>Pseudomonas aeruginosa</i> Elastase LasB by Virgyl Camberlein, Gwenaëlle Jézéquel, Jörg Haupenthal, Anna K. H. Hirsch

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The effects of nifedipine on respiratory mechanics investigated by theend-inflation occlusion method in the rat by Alessandro Rubini, Vincenzo Catena, Daniele del Monte, Gerardo Bosco

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Inhibition of acetylcholinesterase and butyrylcholinesterase with uracil derivatives: kinetic and computational studies by Huseyin Cavdar, Murat Senturk, Murat Guney, Serdar Durdagi, Gulru Kayik, Claudiu T. Supuran, Deniz Ekinci

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Antimicrobial metal-based thiophene derived compounds by Shakeela Yasmeen, Sajjad Hussain Sumrra, Muhammad Safwan Akram, Zahid H. Chohan

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