Search Results - "Medicinal Chemistry"

Tetrahydroquinazole-based secondary sulphonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IV, and IX, and computational studies by Emma Baglini, Rahul Ravichandran, Emanuela Berrino, Silvia Salerno, Elisabetta Barresi, Anna Maria Marini, Monica Viviano, Sabrina Castellano, Federico Da Settimo, Claudiu T. Supuran, Sandro Cosconati, Sabrina Taliani

Connect to this object online.

Design, synthesis and anticancer activity of naphthoquinone derivatives by Xiao-bao Shen, Yang Wang, Xuan-zhen Han, Liang-quan Sheng, Fu-fang Wu, Xinhua Liu

Connect to this object online.

A nanobody-derived mimotope against VEGF inhibits cancer angiogenesis by Elmira Karami, Jean-Marc Sabatier, Mahdi Behdani, Shiva Irani, Fatemeh Kazemi-Lomedasht

Connect to this object online.

Structural/Functional Matches and Divergences of Phytoprostanes and Phytofurans with Bioactive Human Oxylipins by Sonia Medina, Ángel Gil-Izquierdo, Thierry Durand, Federico Ferreres, Raúl Domínguez-Perles

Connect to this object online.

A Narrative Review of Benzo-Fused Coumarins, Shedding Light on Their Medicinal Activities by Yasser Mustafa, Sarah Waheed, Sara Jasim, Rahma Jebir, Reem Ismael, Omar Qutachi

Connect to this object online.

DNA topoisomerases as molecular targets for anticancer drugs by Kamila Buzun, Anna Bielawska, Krzysztof Bielawski, Agnieszka Gornowicz

Connect to this object online.

Synthesis and biological evaluation of 3-arylbenzofuranone derivatives as potential anti-Alzheimer's disease agents by Jie Yang, Yinling Yun, Yuhang Miao, Jie Sun, Xiaojing Wang

Connect to this object online.

PROTACs for BRDs proteins in cancer therapy: a review by Chao Wang, Yujing Zhang, Shanbo Yang, Wujun Chen, Dongming Xing

Connect to this object online.

Of mitochondrion and COVID-19 by Khalid Omer Alfarouk, Sari T. S. Alhoufie, Abdelhameed Hifny, Laurent Schwartz, Ali S. Alqahtani, Samrein B. M. Ahmed, Ali M. Alqahtani, Saad S. Alqahtani, Abdel Khalig Muddathir, Heyam Ali, Adil H. H. Bashir, Muntaser E. Ibrahim, Maria Raffaella Greco, Rosa A. Cardone, Salvador Harguindey, Stephan Joel Reshkin

Connect to this object online.

Exploration of the residues modulating the catalytic features of human carbonic anhydrase XIII by a site-specific mutagenesis approach by Giuseppina De Simone, Anna Di Fiore, Emanuela Truppo, Emma Langella, Daniela Vullo, Claudiu T. Supuran, Simona Maria Monti

Connect to this object online.

Determination of the inhibitory effects of N-methylpyrrole derivatives on glutathione reductase enzyme by Esma Kocaoğlu, Oktay Talaz, Hüseyin Çavdar, Murat Şentürk, Claudiu T. Supuran, Deniz Ekinci

Connect to this object online.

The design, synthesis and antiplasmodial evaluation of novel sulfoximine-isoxazole hybrids as potential antimalarial agents by Jackie L. Mabasa, Tommy F. Mabasa, Musawenkosi L. Nyathi, Paseka T. Moshapo

Connect to this object online.

Can Immobilized Artificial Membrane Chromatography Support the Characterization of Antimicrobial Peptide Origin Derivatives? by Krzesimir Ciura, Natalia Ptaszyńska, Hanna Kapica, Monika Pastewska, Anna Łęgowska, Krzysztof Rolka, Wojciech Kamysz, Wiesław Sawicki, Katarzyna E. Greber

Connect to this object online.

Fragment-pair based drug molecule solubility prediction through attention mechanism by Jianping Liu, Xiujuan Lei, Chunyan Ji, Yi Pan, Yi Pan

Connect to this object online.

Synthesis and biological evaluation of novel thienopyrimidine derivatives as diacylglycerol acyltransferase 1 (DGAT-1) inhibitors by Dong Jin Hong, Seung Hyun Jung, Jisook Kim, Danbee Jung, Young Gil Ahn, Kwee Hyun Suh, Kyung Hoon Min

Connect to this object online.

Carbonic anhydrases from Trypanosoma cruzi and Leishmania donovani chagasi are inhibited by benzoxaboroles by Alessio Nocentini, Roberta Cadoni, Pascal Dumy, Claudiu T. Supuran, Jean-Yves Winum

Connect to this object online.

Arylsulfonamido-alkyl-sulfamates act as inhibitors of bovine carbonic anhydrase II by Toni C. Denner, Niels V. Heise, René Csuk

Connect to this object online.

Sulfur - fluorine bond in PET radiochemistry by Giancarlo Pascali, Lidia Matesic, Bo Zhang, Andrew T. King, Andrea J. Robinson, Alison T. Ung, Benjamin H. Fraser

Connect to this object online.

Research progress of coumarins and their derivatives in the treatment of diabetes by Yinbo Pan, Teng Liu, Xiaojing Wang, Jie Sun

Connect to this object online.

Synthesis and biological evaluation of stilbene derivatives coupled to NO donors as potential antidiabetic agents by Bing Wang, Teng Liu, Zhongyu Wu, Lei Zhang, Jie Sun, Xiaojing Wang

Connect to this object online.