Search Results - "Medicinal Chemistry"

Characterisation of naturally occurring isothiocyanates as glutathione reductase inhibitors by Xia Li, Maowei Ni, Xiaoling Xu, Wei Chen

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Beta-lactamase database (BLDB) - structure and function by Thierry Naas, Saoussen Oueslati, Rémy A. Bonnin, Maria Laura Dabos, Agustin Zavala, Laurent Dortet, Pascal Retailleau, Bogdan I. Iorga

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High-throughput discovery of novel small-molecule inhibitors of acid Ceramidase by Mazen Aseeri, José Luis Abad, Antonio Delgado, Gemma Fabriàs, Gemma Triola, Josefina Casas

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Discovery of (phenylureido)piperidinyl benzamides as prospective inhibitors of bacterial autolysin E from Staphylococcus aureus by Jure Borišek, Sara Pintar, Mitja Ogrizek, Simona Golič Grdadolnik, Vesna Hodnik, Dušan Turk, Andrej Perdih, Marjana Novič

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Medicinal polypharmacology-a scientific glossary of terminology and concepts by Sven Marcel Stefan, Sven Marcel Stefan, Muhammad Rafehi, Muhammad Rafehi

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3-aryl-4-(3,4,5-trimethoxyphenyl)pyridines inhibit tubulin polymerisation and act as anticancer agents by Chao Wang, Yujing Zhang, Shanbo Yang, Lingyu Shi, Yutao Xiu, Yudong Wu, Hongfei Jiang

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Development of novel ALOX15 inhibitors combining dual machine learning filtering and fragment substitution optimisation approaches, molecular docking and dynamic simulation methods by Yinglin Liao, Peng Cao, Lianxiang Luo

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Design, synthesis, molecular dynamics studies and biological evaluations of 4-hydroxy-5-pyrrolinone-3-carbohydrazides as HIV-1 integrase inhibitors by Nafiseh Karimi, Amirreza Dowlati Beirami, Rouhollah Vahabpour Roudsari, Zahra Hajimahdi, Afshin Zarghi

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Synthetic marvels in tuberculosis research: An in-depth review of 1,3,4-oxadiazole derivatives as antitubercular agents by Isha Kapila, Ankita Bharwal, Poonam Sharma, Neeraj Choudhary, Vikrant Abbot

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Structure-based design of ligands of the m6A-RNA reader YTHDC1 by Yaozong Li, Rajiv Kumar Bedi, Francesco Nai, Valentin von Roten, Aymeric Dolbois, František Zálešák, Raed Nachawati, Danzhi Huang, Amedeo Caflisch

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Tyrosinase inhibitory components from Aloe vera and their antiviral activity by Jang Hoon Kim, Ju-Yeon Yoon, Seo Young Yang, Seung-Kook Choi, Sun Jung Kwon, In Sook Cho, Min Hee Jeong, Young Ho Kim, Gug Seoun Choi

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Anticancer sulfonamide hybrids that inhibit bladder cancer cells growth and migration as tubulin polymerisation inhibitors by Jia Liu, Chunlai Liu, Xiling Zhang, Liu Yu, Xue Gong, Ping Wang

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Macrocarpal C isolated from Eucalyptus globulus inhibits dipeptidyl peptidase 4 in an aggregated form by Eisuke Kato, Kazuhiro Kawakami, Jun Kawabata

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Paving the way towards effective plant-based inhibitors of hyaluronidase and tyrosinase: a critical review on a structure-activity relationship by Jakub Gębalski, Filip Graczyk, Daniel Załuski

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Discovery of new chromen-4-one derivatives as telomerase inhibitors through regulating expression of dyskerin by Jie Quan Wang, Meng Di Yang, Xing Chen, Yang Wang, Liu Zeng Chen, Xiu Cheng, Xin Hua Liu

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Exploring new structural features of the 4-[(3-methyl-4-aryl-2,3-dihydro-1,3-thiazol-2-ylidene)amino]benzenesulphonamide scaffold for the inhibition of human carbonic anhydrases by Simona Distinto, Rita Meleddu, Francesco Ortuso, Filippo Cottiglia, Serenella Deplano, Lisa Sequeira, Claudia Melis, Benedetta Fois, Andrea Angeli, Clemente Capasso, Rossella Angius, Stefano Alcaro, Claudiu T. Supuran, Elias Maccioni

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Kushenol A and 8-prenylkaempferol, tyrosinase inhibitors, derived from Sophora flavescens by Jang Hoon Kim, In Sook Cho, Yang Kang So, Hyeong-Hwan Kim, Young Ho Kim

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Statins interfere with the attachment of S. cerevisiae mtDNA to the inner mitochondrial membrane by Angela Cirigliano, Antonia Amelina, Beatrice Biferali, Alberto Macone, Chiara Mozzetta, Michele Maria Bianchi, Mattia Mori, Bruno Botta, Elah Pick, Rodolfo Negri, Teresa Rinaldi

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Styrylquinazoline derivatives as ABL inhibitors selective for different DFG orientations by Katarzyna Malarz, Jacek Mularski, Marcin Pacholczyk, Robert Musiol

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Design and synthesis of a novel photoaffinity probe for labelling EGF receptor tyrosine kinases by You-Guang Zheng, Xiao-Qing Wu, Jun Su, Ping Jiang, Liang Xu, Jian Gao, Bin Cai, Min Ji

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