Search Results - "Medicinal Chemistry"

Novel group of tyrosyl-DNA-phosphodiesterase 1 inhibitors based on disaccharide nucleosides as drug prototypes for anti-cancer therapy by Anastasia O. Komarova, Mikhail S. Drenichev, Nadezhda S. Dyrkheeva, Irina V. Kulikova, Vladimir E. Oslovsky, Olga D. Zakharova, Alexandra L. Zakharenko, Sergey N. Mikhailov, Olga I. Lavrik

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Inhibition of bacterial and human zinc-metalloproteases by bisphosphonate- and catechol-containing compounds by Fatema Rahman, Tra-Mi Nguyen, Olayiwola A. Adekoya, Cristina Campestre, Paolo Tortorella, Ingebrigt Sylte, Jan-Olof Winberg

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Different roles for the acyl chain and the amine leaving group in the substrate selectivity of N-Acylethanolamine acid amidase by Andrea Ghidini, Laura Scalvini, Francesca Palese, Alessio Lodola, Marco Mor, Daniele Piomelli

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Latest advances in dual inhibitors of acetylcholinesterase and monoamine oxidase B against Alzheimer's disease by Dajiang Zou, Renzheng Liu, Yangjing Lv, Jianan Guo, Changjun Zhang, Yuanyuan Xie

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Dithiocarbamates effectively inhibit the α-carbonic anhydrase from Neisseria gonorrhoeae by Simone Giovannuzzi, Nader S. Abutaleb, Chad S. Hewitt, Fabrizio Carta, Alessio Nocentini, Mohamed N. Seleem, Daniel P. Flaherty, Claudiu T. Supuran

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A new colorimetric DPPH• scavenging activity method with no need for a spectrophotometer applied on synthetic and natural antioxidants and medicinal herbs by Zeynep Akar, Murat Küçük, Hacer Doğan

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Discovering a new class of antifungal agents that selectively inhibits microbial carbonic anhydrases by Giannamaria Annunziato, Laura Giovati, Andrea Angeli, Marialaura Pavone, Sonia Del Prete, Marco Pieroni, Clemente Capasso, Agostino Bruno, Stefania Conti, Walter Magliani, Claudiu T. Supuran, Gabriele Costantino

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Inhibition of soluble epoxide hydrolase by phytochemical constituents of the root bark of Ulmus davidiana var. japonica by Jang Hoon Kim, Ji Su Park, Yun Ji Lee, Sena Choi, Young Ho Kim, Seo Young Yang

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Impact of phytosterols on liver and distal colon metabolome in experimental murine colitis model: an explorative study by Nunzia Iaccarino, Jussara Amato, Bruno Pagano, Anna Di Porzio, Matteo Micucci, Luca Bolelli, Rita Aldini, Ettore Novellino, Roberta Budriesi, Antonio Randazzo

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Synthesis and biological evaluation of aminomethyl and alkoxymethyl derivatives as carbonic anhydrase, acetylcholinesterase and butyrylcholinesterase inhibitors by İlhami Gulçin, Malahat Abbasova, Parham Taslimi, Zübeyir Huyut, Leyla Safarova, Afsun Sujayev, Vagif Farzaliyev, Şükrü Beydemir, Saleh H. Alwasel, Claudiu T. Supuran

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Pharmaceutical strategies for preventing toxicity and promoting antioxidant and anti-inflammatory actions of bilirubin by Alessio Nocentini, Alessandro Bonardi, Simone Pratesi, Paola Gratteri, Carlo Dani, Claudiu T. Supuran

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Synthesis and biological evaluation of anti-Toxoplasma gondii activity of a novel scaffold of thiazolidinone derivatives by Simone Carradori, Daniela Secci, Bruna Bizzarri, Paola Chimenti, Celeste De Monte, Paolo Guglielmi, Cristina Campestre, Daniela Rivanera, Claudia Bordón, Lorraine Jones-Brando

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Design, synthesis, and biological evaluation of piperazine derivatives involved in the 5-HT1AR/BDNF/PKA pathway by Hao Zhou, Mengjiao Li, Hui Liu, Zheng Liu, Xuekun Wang, Shiben Wang

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Antimycobacterial activity of nitrogen heterocycles derivatives: 7-(pyridine-4-yl)-indolizine derivatives. Part VII8-12 by Anda-Mihaela Olaru, Violeta Vasilache, Ramona Danac, Ionel I. Mangalagiu

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Identification and characterization of the α-CA in the outer membrane vesicles produced by Helicobacter pylori by Maurizio Ronci, Sonia Del Prete, Valentina Puca, Simone Carradori, Vincenzo Carginale, Raffaella Muraro, Gabriella Mincione, Antonio Aceto, Francesca Sisto, Claudiu T. Supuran, Rossella Grande, Clemente Capasso

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Novel tyrosinase inhibitory peptide with free radical scavenging ability by Zhiwei Shen, Yujiao Wang, Zhen Guo, Tingyuan Tan, Yi Zhang

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Assessment of Anti-tyrosinase and Antioxidant Activities along with Molecular Docking Studies, and in silico ADME of Some 3-Hydroxypyridin-4-one Derivatives by Fateme Zare, Sara Sadeghian, Mehdi Khoshneviszadeh, Mojgan Pasbani, Razieh Sabet, Hossein Sadeghpour

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Rosmarinic acid prevents fibrillization and diminishes vibrational modes associated to β sheet in tau protein linked to Alzheimer's disease by Alberto Cornejo, Felipe Aguilar Sandoval, Leonardo Caballero, Luis Machuca, Patricio Muñoz, Julio Caballero, George Perry, Alejandro Ardiles, Carlos Areche, Francisco Melo

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Discovery of 3-alkyl-5-aryl-1-pyrimidyl-1H-pyrazole derivatives as a novel selective inhibitor scaffold of JNK3 by Youri Oh, Miyoung Jang, Hyunwook Cho, Songyi Yang, Daseul Im, Hyungwoo Moon, Jung-Mi Hah

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Reversal of Multidrug Resistance by Symmetrical Selenoesters in Colon Adenocarcinoma Cells by Bálint Rácz, Annamária Kincses, Krisztián Laczi, Gábor Rákhely, Enrique Domínguez-Álvarez, Gabriella Spengler

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