Search Results - "Medicinal Chemistry"

Quantitative assessment of specific carbonic anhydrase inhibitors effect on hypoxic cells using electrical impedance assays by Luciana Stanica, Mihaela Gheorghiu, Miruna Stan, Cristina Polonschii, Sorin David, Dumitru Bratu, Anca Dinischiotu, Claudiu T. Supuran, Eugen Gheorghiu

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An anion and small molecule inhibition study of the β-carbonic anhydrase from Staphylococcus aureus by Linda J. Urbanski, Daniela Vullo, Seppo Parkkila, Claudiu T. Supuran

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The new H2S-releasing compound ACS94 exerts protective effects through the modulation of thiol homoeostasis by Daniela Giustarini, Valerio Tazzari, Ivan Bassanini, Ranieri Rossi, Anna Sparatore

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Anilino-1,4-naphthoquinones as potent mushroom tyrosinase inhibitors: in vitro and in silico studies by Sahachai Sabuakham, Sutita Nasoontorn, Napat Kongtaworn, Thanyada Rungrotmongkol, Atit Silsirivanit, Ratchanok Pingaew, Panupong Mahalapbutr

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Aryl derivatives of 3H-1,2-benzoxaphosphepine 2-oxides as inhibitors of cancer-related carbonic anhydrase isoforms IX and XII by Anastasija Balašova, Aleksandrs Pustenko, Alessio Nocentini, Daniela Vullo, Claudiu T. Supuran, Raivis Žalubovskis

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Prostate cancer cells and exosomes in acidic condition show increased carbonic anhydrase IX expression and activity by Mariantonia Logozzi, Clemente Capasso, Rossella Di Raimo, Sonia Del Prete, Davide Mizzoni, Mario Falchi, Claudiu T. Supuran, Stefano Fais

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Charged pyridinium oximes with thiocarboxamide moiety are equally or less effective reactivators of organophosphate-inhibited cholinesterases compared to analogous carboxamides by Zuzana Kohoutova, David Malinak, Rudolf Andrys, Jana Svobodova, Miroslav Psotka, Monika Schmidt, Lukas Prchal, Kamil Musilek

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3D QSAR studies, pharmacophore modeling, and virtual screening of diarylpyrazole-benzenesulfonamide derivatives as a template to obtain new inhibitors, using human carbonic anhydra... by Yeganeh Entezari Heravi, Hassan Sereshti, Ali Akbar Saboury, Jahan Ghasemi, Marzieh Amirmostofian, Claudiu T. Supuran

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Recent progress in chemistry and bioactivity of monoterpenoid indole alkaloids from the genus gelsemium: a comprehensive review by Lin Wang, Siyu Chen, Xun Gao, Xiao Liang, Weichen Lv, Dongfang Zhang, Xin Jin

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Synthesis and structure-activity relationships of novel 5-(hydroxamic acid)methyl oxazolidinone derivatives as 5-lipoxygenase inhibitors by Oludotun A. Phillips, Mira A. Bosso, Charles I. Ezeamuzie

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Benzylamides and piperazinoarylamides of ibuprofen as fatty acid amide hydrolase inhibitors by Alessandro Deplano, Mariateresa Cipriano, Federica Moraca, Ettore Novellino, Bruno Catalanotti, Christopher J. Fowler, Valentina Onnis

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Development of potent reversible selective inhibitors of butyrylcholinesterase as fluorescent probes by Stane Pajk, Damijan Knez, Urban Košak, Maja Zorović, Xavier Brazzolotto, Nicolas Coquelle, Florian Nachon, Jacques-Philippe Colletier, Marko Živin, Jure Stojan, Stanislav Gobec

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Novel positive allosteric modulators of A2B adenosine receptor acting as bone mineralisation promoters by Elisabetta Barresi, Chiara Giacomelli, Laura Marchetti, Emma Baglini, Silvia Salerno, Giovanni Greco, Federico Da Settimo, Claudia Martini, Maria Letizia Trincavelli, Sabrina Taliani

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Effects of thymoquinone and the curcumin analog EF-24 on the activity of the enzyme paraoxonase-1 in human glioblastoma cells U87MG by Ender Simsek, Asuman Sunguroglu, Ahmet Kilic, Nurbanu Özgültekin, O. Ozensoy Guler

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Design, synthesis and in vitro antiproliferative activity of new thiazolidinedione-1,3,4-oxadiazole hybrids as thymidylate synthase inhibitors by Zohor Mohammad Mahdi Alzhrani, Mohammad Mahboob Alam, Thikryat Neamatallah, Syed Nazreen

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Searching for drug leads targeted to the hydrophobic cleft of dengue virus capsid protein by Liliane O. Ortlieb, Ícaro P. Caruso, Nathane C. Mebus-Antunes, Andrea T. Da Poian, Elaine da C. Petronilho, José Daniel Figueroa-Villar, Claudia J. Nascimento, Fabio C. L. Almeida

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α-Glucosidase inhibition by flavonoids: an in vitro and in silico structure-activity relationship study by Carina Proença, Marisa Freitas, Daniela Ribeiro, Eduardo F. T. Oliveira, Joana L. C. Sousa, Sara M. Tomé, Maria J. Ramos, Artur M. S. Silva, Pedro A. Fernandes, Eduarda Fernandes

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Synthesis, antimycobacterial evaluation, and molecular docking study of 1,2,4-triazole derivatives by Meng-Yu Xia, Yu-Xiang Cai, Jun-Xian Chen, Xin Zhao, Hong-Mei Dong, Zai-Chang Yang

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Determination and diagnostic value of CA9 mRNA in peripheral blood of patients with oral leukoplakia by Manuel Torres López, Mario Pérez Sayáns, Cintia Chamorro Petronacci, Francisco Barros Angueira, Pilar Gándara Vila, Alejandro Lorenzo Pouso, Abel García García

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Activation studies with amino acids and amines of a β-carbonic anhydrase from Mammaliicoccus (Staphylococcus) sciuri previously annotated as Staphylococcus aureus (SauBCA) carbonic... by Andrea Angeli, Linda J Urbański, Clemente Capasso, Seppo Parkkila, Claudiu T. Supuran

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