Search Results - "Medicinal Chemistry"

Two approaches to the use of benzo[c][1,2]oxaboroles as active fragments for synthetic transformation of clarithromycin by Gennady B. Lapa, Elena P. Mirchink, Elena B Isakova, Maria N Preobrazhenskaya

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Inhibition studies of Brucella suis β-carbonic anhydrases with a series of 4-substituted pyridine-3-sulphonamides by Simona Maria Monti, Angela Meccariello, Mariangela Ceruso, Krzysztof Szafrański, Jarosław Sławiński, Claudiu T. Supuran

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HPLC-UV assay for the evaluation of inhibitors of plasma amine oxidase using crude bovine plasma by Kira Mergemeier, Florian Galster, Matthias Lehr

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Resolution of co-eluting isomers of anti-inflammatory drugs conjugated to carbonic anhydrase inhibitors from plasma in liquid chromatography by energy-resolved tandem mass spectrom... by Marta Menicatti, Marco Pallecchi, Silvia Bua, Daniela Vullo, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Fabrizio Carta, Claudiu T. Supuran, Gianluca Bartolucci

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Novel piperidine derivatives as colchicine binding site inhibitors induce apoptosis and inhibit epithelial-mesenchymal transition against prostate cancer PC3 cells by Dong-Jun Fu, Si-Meng Liu, Jia-Jia Yang, Jun Li

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Assessment of the antiproliferative and apoptotic roles of sulfonamide carbonic anhydrase IX inhibitors in HeLa cancer cell line by Ismail Koyuncu, Ataman Gonel, Mustafa Durgun, Abdurrahim Kocyigit, Ozgur Yuksekdag, Claudiu T. Supuran

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Development of novel anilinoquinazoline-based carboxylic acids as non-classical carbonic anhydrase IX and XII inhibitors by Zainab M. Elsayed, Hadia Almahli, Alessio Nocentini, Andrea Ammara, Claudiu T. Supuran, Wagdy M. Eldehna, Sahar M. Abou-Seri

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Inhibition studies with simple and complex (in)organic anions of the γ-carbonic anhydrase from Mammaliicoccus (Staphylococcus) sciuri, MscCAγ by Simone Giovannuzzi, Viviana De Luca, Clemente Capasso, Claudiu T. Supuran

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Inhibition potential of phenolic constituents from the aerial parts of Tetrastigma hemsleyanum against soluble epoxide hydrolase and nitric oxide synthase by Cai Yi Wang, Sunggun Lee, Hyun-Jae Jang, Xiang Dong Su, Heng-Shan Wang, Young Ho Kim, Seo Young Yang

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Pterostilbene fluorescent probes as potential tools for targeting neurodegeneration in biological applications by Lidia Ciccone, Susanna Nencetti, Maria Marino, Chiara Battocchio, Giovanna Iucci, Iole Venditti, Martina Marsotto, Emiliano Montalesi, Simone Socci, Beatrice Bargagna, Elisabetta Orlandini

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Analogues of 2'-hydroxychalcone with modified C4-substituents as the inhibitors against human acetylcholinesterase by Sri Devi Sukumaran, Shah Bakhtiar Nasir, Jia Ti Tee, Michael J. C. Buckle, Rozana Othman, Noorsaadah Abd. Rahman, Vannajan Sanghiran Lee, Syed Nasir Abbas Bukhari, Chin Fei Chee

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Synthesis and biological evaluation of histamine Schiff bases as carbonic anhydrase I, II, IV, VII, and IX activators by Suleyman Akocak, Nabih Lolak, Daniela Vullo, Mustafa Durgun, Claudiu T. Supuran

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CO2 permeability of the rat erythrocyte membrane and its inhibition by Samer Al-Samir, Maximilian Prill, Claudiu T. Supuran, Gerolf Gros, Volker Endeward

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Unveiling the mechanism of action of acylated temporin L analogues against multidrug-resistant Candida albicans by Rosa Bellavita, Annarita Falanga, Francesco Merlino, Gabriella D'Auria, Nicola Molfetta, Anella Saviano, Francesco Maione, Umberto Galdiero, Maria Rosaria Catania, Stefania Galdiero, Paolo Grieco, Emanuela Roscetto, Lucia Falcigno, Elisabetta Buommino

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Boronic acid inhibitors of penicillin-binding protein 1b: serine and lysine labelling agents by Levente Kollár, Katarina Grabrijan, Martina Hrast Rambaher, Krištof Bozovičar, Tímea Imre, György G. Ferenczy, Stanislav Gobec, György M. Keserű

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Design, synthesis and docking study of novel coumarin ligands as potential selective acetylcholinesterase inhibitors by Fatih Sonmez, Belma Zengin Kurt, Isil Gazioglu, Livia Basile, Aydan Dag, Valentina Cappello, Tiziana Ginex, Mustafa Kucukislamoglu, Salvatore Guccione

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Bio-inspired green fabrication of silver nanoparticles (AgNPs) using aqueous leaves extract of Ipomoea carnea Jacq. To tackle multiple drug resistance MTCC bacterial strains by Ramveer Singh, Narashans Alok Sagar, Navneet Kumar

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Nanovesicles released by OKT3 hybridoma express fully active antibodies by Mariantonia Logozzi, Rossella Di Raimo, Francesca Properzi, Stefano Barca, Daniela F. Angelini, Davide Mizzoni, Mario Falchi, Luca Battistini, Stefano Fais

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Design, synthesis and biological evaluation of a series of dianilinopyrimidines as EGFR inhibitors by Longjia Yan, Qin Wang, Li Liu, Yi Le

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Repurposing of rabeprazole as an anti-Trypanosoma cruzi drug that targets cellular triosephosphate isomerase by Itzhel García-Torres, Ignacio De la Mora-De la Mora, Gabriel López-Velázquez, Nallely Cabrera, Luis Antonio Flores-López, Ingeborg Becker, Juliana Herrera-López, Roberto Hernández, Ruy Pérez-Montfort, Sergio Enríquez-Flores

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