Search Results - "Medicinal Chemistry"

Design and synthesis of new spirooxindole candidates and their selenium nanoparticles as potential dual Topo I/II inhibitors, DNA intercalators, and apoptotic inducers by Samar El-Kalyoubi, Mohamed M. Khalifa, Mahmoud T. Abo-Elfadl, Ahmed A. El-Sayed, Ahmed Elkamhawy, Kyeong Lee, Ahmed A. Al-Karmalawy

Connect to this object online.

A novel RRGW derived peptide is a promising inhibitor of BoNT/A by Wantong Ma, Lulu Wang, Xiangmin Tan, Xin Wang, Chunyan Yang, Yu Wang, Ziye Liu, Bo Liu, Hai Zhu, Dejuan Zhi, Dongsheng Wang

Connect to this object online.

Quinoline Derivatives: Promising Antioxidants with Neuroprotective Potential by Luis Felipe Hernández-Ayala, Eduardo Gabriel Guzmán-López, Annia Galano

Connect to this object online.

Multicomponent pattern and biological activities of seven Asphodeline taxa: potential sources of natural-functional ingredients for bioactive formulations by Marcello Locatelli, Gokhan Zengin, Ahmet Uysal, Simone Carradori, Elisa De Luca, Giuseppe Bellagamba, Abdurrahman Aktumsek, Irina Lazarova

Connect to this object online.

Phosphorus containing analogues of SAHA as inhibitors of HDACs by Michael D. Pun, Hsin-Hua Wu, Feyisola P. Olatunji, Britany N. Kesic, John W. Peters, Clifford E. Berkman

Connect to this object online.

Metallo-antiviral aspirants: Answer to the upcoming virus outbreak by Ripul Mehrotra, Satyendra N. Shukla, Pratiksha Gaur

Connect to this object online.

Structure-guided discovery of novel dUTPase inhibitors with anti-Nocardia activity by computational design by Zhi-Zheng Wang, Jun Weng, Jing Qi, Xin-Xin Fu, Ban-Bin Xing, Yang Hu, Chun-Hsiang Huang, Chin-Yu Chen, Zigong Wei

Connect to this object online.

Synthesis and Atimicrobial Evaluation of Deuterated Analogues of Metronidazole by Anjana G V

Connect to this object online.

8-Mercaptoguanine-based inhibitors of Mycobacterium tuberculosis dihydroneopterin aldolase: synthesis, in vitro inhibition and docking studies by Alexia de Matos Czeczot, Candida Deves Roth, Rodrigo Gay Ducati, Kenia Pissinate, Raoní Scheibler Rambo, Luís Fernando Saraiva Macedo Timmers, Bruno Lopes Abbadi, Fernanda Souza Macchi, Víctor Zajaczkowski Pestana, Luiz Augusto Basso, Pablo Machado, Cristiano Valim Bizarro

Connect to this object online.

Discovery of a novel Aurora B inhibitor GSK650394 with potent anticancer and anti-aspergillus fumigatus dual efficacies in vitro by Yuhua He, Wei Fu, Liyang Du, Huiqiao Yao, Zhengkang Hua, Jinyu Li, Zhonghui Lin

Connect to this object online.

Flavone-based dual PARP-Tubulin inhibitor manifesting efficacy against endometrial cancer by Sachin Sharma, Kavya Chandra, Aliva Naik, Anamika Sharma, Ram Sharma, Amandeep Thakur, Ajmer Singh Grewal, Ashwani K. Dhingra, Arnab Banerjee, Jing Ping Liou, Santosh Kumar Guru, Kunal Nepali

Connect to this object online.

Inhibition of Shiga toxin-converting bacteriophage development by novel antioxidant compounds by Sylwia Bloch, Bożena Nejman-Faleńczyk, Karolina Pierzynowska, Ewa Piotrowska, Alicja Węgrzyn, Christelle Marminon, Zouhair Bouaziz, Pascal Nebois, Joachim Jose, Marc Le Borgne, Luciano Saso, Grzegorz Węgrzyn

Connect to this object online.

Design and synthesis of naphthalimide group-bearing thioglycosides as novel β-N-acetylhexosaminidases inhibitors by Shengqiang Shen, Wei Chen, Lili Dong, Qing Yang, Huizhe Lu, Jianjun Zhang

Connect to this object online.

The lignicolous fungus Trametes versicolor (L.) Lloyd (1920): a promising natural source of antiradical and AChE inhibitory agents by Ljiljana Janjušević, Maja Karaman, Filip Šibul, Giuseppina Tommonaro, Carmine Iodice, Dragica Jakovljević, Boris Pejin

Connect to this object online.

Benzimidazole-based derivatives as privileged scaffold developed for the treatment of the RSV infection: a computational study exploring the potency and cytotoxicity profiles by Elena Cichero, Michele Tonelli, Federica Novelli, Bruno Tasso, Ilenia Delogu, Roberta Loddo, Olga Bruno, Paola Fossa

Connect to this object online.

Pyrrolo[3,2-c]pyridine derivatives with potential inhibitory effect against FMS kinase: in vitro biological studies by Mohammed I. El-Gamal, Chang-Hyun Oh

Connect to this object online.

HT-SuMD: making molecular dynamics simulations suitable for fragment-based screening. A comparative study with NMR by Francesca Ferrari, Maicol Bissaro, Simone Fabbian, Jessica De Almeida Roger, Stefano Mammi, Stefano Moro, Massimo Bellanda, Mattia Sturlese

Connect to this object online.

Protective effects of carbonic anhydrase inhibition in brain ischaemia in vitro and in vivo models by Ilaria Dettori, Irene Fusco, Irene Bulli, Lisa Gaviano, Elisabetta Coppi, Federica Cherchi, Martina Venturini, Lorenzo Di Cesare Mannelli, Carla Ghelardini, Alessio Nocentini, Claudiu T. Supuran, Anna Maria Pugliese, Felicita Pedata

Connect to this object online.

Synthesis and biological evaluation of 4-phenoxy-phenyl isoxazoles as novel acetyl-CoA carboxylase inhibitors by Xin Wu, Yongbo Yu, Tonghui Huang

Connect to this object online.

4-Cyanamidobenzenesulfonamide derivatives: a novel class of human and bacterial carbonic anhydrase inhibitors by Morteza Abdoli, Alessandro Bonardi, Claudiu T. Supuran, Raivis Žalubovskis

Connect to this object online.