Search Results - "Medicinal Chemistry"

Interactions of 2,6-substituted purines with purine nucleoside phosphorylase from Helicobacter pylori in solution and in the crystal, and the effects of these compounds on cell cul... by Marta Narczyk, Marta Ilona Wojtyś, Ivana Leščić Ašler, Biserka Žinić, Marija Luić, Elżbieta Katarzyna Jagusztyn-Krynicka, Zoran Štefanić, Agnieszka Bzowska

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Synthesis, computational studies and assessment of in vitro inhibitory activity of umbelliferon-based compounds against tumour-associated carbonic anhydrase isoforms IX and XII by Francesca Mancuso, Laura De Luca, Andrea Angeli, Sonia Del Prete, Clemente Capasso, Claudiu T. Supuran, Rosaria Gitto

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SYNTHESIS AND PHARMACOLOGICAL EVALUATION: ANTIMICROBIAL, ANTI-INFLAMMATORY, ANALGESIC, ULCEROGENIC PROPERTIES OF SEVERAL BIS-HETEROCYCLIC DERIVATIVES by Ravindra Kumar, Hament Panwar

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Coumarins from Magydaris pastinacea as inhibitors of the tumour-associated carbonic anhydrases IX and XII: isolation, biological studies and in silico evaluation by Benedetta Fois, Simona Distinto, Rita Meleddu, Serenella Deplano, Elias Maccioni, Costantino Floris, Antonella Rosa, Mariella Nieddu, Pierluigi Caboni, Claudia Sissi, Andrea Angeli, Claudiu T. Supuran, Filippo Cottiglia

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Evaluation of N-alkyl isatins and indoles as acetylcholinesterase and butyrylcholinesterase inhibitors by Kaitlyn N. Alcorn, Isabelle A. Oberhauser, Matthew D. Politeski, Todd J. Eckroat

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Microtiter plate-based chemistry and in situ screening: SuFEx-enabled lead discovery of selective AChE inhibitors by Kun Tang, Huan-Huan Li, Chengyao Wu, Shi-Long Zhang, Jian-Guo Yang, Wenjian Tang, Hua-Li Qin

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Biochemical and structural characterisation of a protozoan beta-carbonic anhydrase from Trichomonas vaginalis by Linda J. Urbański, Anna Di Fiore, Latifeh Azizi, Vesa P. Hytönen, Marianne Kuuslahti, Martina Buonanno, Simona M. Monti, Andrea Angeli, Reza Zolfaghari Emameh, Claudiu T. Supuran, Giuseppina De Simone, Seppo Parkkila

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Adiponectin - stratification biomarker in diastolic cardiac dysfunction by Valeriu-Gabi Dincă, Adriana Diaconu, Bogdan-Ioan Coculescu, Alexandra-Ligia Dincă, Diana Mihaela Ciuc, Rodica Daniela Bîrlă, Cristian Daniel Marica, Sorin Ioan Tudorache, Gheorghe Manole, Elena Claudia Coculescu

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Discovery of antimicrobial compounds targeting bacterial type FAD synthetases by María Sebastián, Ernesto Anoz-Carbonell, Begoña Gracia, Pilar Cossio, José Antonio Aínsa, Isaías Lans, Milagros Medina

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The inhibitory effect of boric acid on hypoxia-regulated tumour-associated carbonic anhydrase IX by Zainab Saad Yusuf, Tugba Kevser Uysal, Ender Simsek, Alessio Nocentini, Sameh Mohamed Osman, Claudiu T. Supuran, Özen Özensoy Güler

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Cover, Content, and Editorial Note from Borneo J Pharm Vol. 6 No. 4 November 2023 by Chief Editor of Borneo J Pharm

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Activation of human α-carbonic anhydrase isoforms I, II, IV and VII with bis-histamine schiff bases and bis-spinaceamine substituted derivatives by Suleyman Akocak, Nabih Lolak, Silvia Bua, Alessio Nocentini, Claudiu T. Supuran

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Effect of amino acids and amines on the activity of the recombinant ι-carbonic anhydrase from the Gram-negative bacterium Burkholderia territorii by Viviana De Luca, Andrea Petreni, Vincenzo Carginale, Andrea Scaloni, Claudiu T. Supuran, Clemente Capasso

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The gram-negative bacterium Escherichia coli as a model for testing the effect of carbonic anhydrase inhibition on bacterial growth by Viviana De Luca, Vincenzo Carginale, Claudiu T. Supuran, Clemente Capasso

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Design, synthesis and molecular docking of novel diarylcyclohexenone and diarylindazole derivatives as tubulin polymerization inhibitors by Riham I. Ahmed, Essam Eldin A. Osman, Fadi M. Awadallah, Samir M. El-Moghazy

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Reconsidering anion inhibitors in the general context of drug design studies of modulators of activity of the classical enzyme carbonic anhydrase by Alessio Nocentini, Andrea Angeli, Fabrizio Carta, Jean-Yves Winum, Raivis Zalubovskis, Simone Carradori, Clemente Capasso, William A. Donald, Claudiu T. Supuran

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Characterization of human S-adenosyl-homocysteine hydrolase in vitro and identification of its potential inhibitors by Weiwei Hao, Yanhua Li, Qiuli Shan, Tian Han, Wencheng Li, Sheng He, Kongkai Zhu, Yumei Li, Xiaojun Tan, Jinsong Gu

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Chemical composition, seasonal variation and antiaging activities of essential oil from Callistemon subulatus leaves growing in Egypt by Omyma Rabie, Heba A. S. El-Nashar, Taghreed A. Majrashi, Tarfah Al‐Warhi, Mahmoud A. El Hassab, Wagdy M. Eldehna, Nada M. Mostafa

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Design and synthesis of some new benzoylthioureido phenyl derivatives targeting carbonic anhydrase enzymes by Mazin A. A. Najm, Walaa R. Mahmoud, Azza T. Taher, Safinaz E-S. Abbas, Fadi M. Awadallah, Heba Abdelrasheed Allam, Daniela Vullo, Claudiu T. Supuran

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Synthesis and evaluation of a large library of nitroxoline derivatives as pancreatic cancer antiproliferative agents by Serena Veschi, Simone Carradori, Laura De Lellis, Rosalba Florio, Davide Brocco, Daniela Secci, Paolo Guglielmi, Mattia Spano, Anatoly P. Sobolev, Alessandro Cama

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