Search Results - "Medicinal Chemistry"

Biological investigation of N-methyl thiosemicarbazones as antimicrobial agents and bacterial carbonic anhydrases inhibitors by Ilaria D'Agostino, Githa Elizabeth Mathew, Paola Angelini, Roberto Venanzoni, Giancarlo Angeles Flores, Andrea Angeli, Simone Carradori, Beatrice Marinacci, Luigi Menghini, Mohamed A. Abdelgawad, Mohammed M. Ghoneim, Bijo Mathew, Claudiu T. Supuran

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Inhibition studies on a panel of human carbonic anhydrases with N1-substituted secondary sulfonamides incorporating thiazolinone or imidazolone-indole tails by Fadi M. Awadallah, Silvia Bua, Walaa R. Mahmoud, Hossam H. Nada, Alessio Nocentini, Claudiu T. Supuran

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Discovery of novel conjugates of quinoline and thiazolidinone urea as potential anti-colorectal cancer agent by Li Xiong, Huan He, Mengmeng Fan, Liping Hu, Fei Wang, Xiaomeng Song, Shengmin Shi, Baohui Qi

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Do CO2 and oxidative stress induce cancer?: a brief study about the evaluation of PON 1, CAT, CA and XO enzyme levels on head and neck cancer patients by Murad Mutlu, M. Hakan Korkmaz, Ender Simsek, Emine Terzi, Beyza Ecem Oz Bedir, Tugba Kevser Uysal, Omer Bayir, Guleser Saylam, Ozen Ozensoy Guler

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Design, synthesis and molecular modelling studies of some pyrazole derivatives as carbonic anhydrase inhibitors by Yazgı Dizdaroglu, Canan Albay, Tayfun Arslan, Abdulilah Ece, Emir A. Turkoglu, Asiye Efe, Murat Senturk, Claudiu T. Supuran, Deniz Ekinci

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Design of selective COX-2 inhibitors in the (aza)indazole series. Chemistry, in vitro studies, radiochemistry and evaluations in rats of a [18F] PET tracer by Jonathan Elie, Johnny Vercouillie, Nicolas Arlicot, Lucas Lemaire, Rudy Bidault, Sylvie Bodard, Christel Hosselet, Jean-Bernard Deloye, Sylvie Chalon, Patrick Emond, Denis Guilloteau, Frédéric Buron, Sylvain Routier

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Discovery of novel dual-active 3-(4-(dimethylamino)phenyl)-7-aminoalcoxy-coumarin as potent and selective acetylcholinesterase inhibitor and antioxidant by Gabriela Alves de Souza, Soraia John da Silva, Catarina de Nigris Del Cistia, Paulo Pitasse-Santos, Lucas de Oliveira Pires, Yulli Moraes Passos, Yraima Cordeiro, Cristiane Martins Cardoso, Rosane Nora Castro, Carlos Mauricio R. Sant'Anna, Arthur Eugen Kümmerle

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An AGT-based protein-tag system for the labelling and surface immobilization of enzymes on E. coli outer membrane by Rosa Merlo, Sonia Del Prete, Anna Valenti, Rosanna Mattossovich, Vincenzo Carginale, Claudiu T. Supuran, Clemente Capasso, Giuseppe Perugino

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Anti-Helicobacter pylori activity of ethoxzolamide by Joyanta K. Modak, Alexandra Tikhomirova, Rebecca J. Gorrell, Mohammad M. Rahman, Despina Kotsanas, Tony M. Korman, Jose Garcia-Bustos, Terry Kwok, Richard L. Ferrero, Claudiu T. Supuran, Anna Roujeinikova

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Methotrexate, an anti-inflammatory drug, inhibits Hepatitis E viral replication by Akash Kumar, Preeti Hooda, Anindita Puri, Radhika Khatter, Mohammed S. Al-Dosari, Neha Sinha, Mohammad K. Parvez, Deepak Sehgal

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Gualou Guizhi decoction reverses brain damage with cerebral ischemic stroke, multi-component directed multi-target to screen calcium-overload inhibitors using combination of molecu... by Juan Hu, Wen-Sheng Pang, Jing Han, Kuan Zhang, Ji-Zhou Zhang, Li-Dian Chen

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An Overview on Patient-Centered Clinical Services by Gaurav Joshi, Atul Kabra, Nishant Goutam, Alka Sharma

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Anti-influenza A virus activity and structure-activity relationship of a series of nitrobenzoxadiazole derivatives by Francesco Fiorentino, Marta De Angelis, Martina Menna, Annarita Rovere, Anna Maria Caccuri, Francesca D'Acunzo, Anna Teresa Palamara, Lucia Nencioni, Dante Rotili, Antonello Mai

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Methoxy and bromo scans on N-(5-methoxyphenyl) methoxybenzenesulphonamides reveal potent cytotoxic compounds, especially against the human breast adenocarcinoma MCF7 cell line by Myriam González, María Ovejero-Sánchez, Alba Vicente-Blázquez, Manuel Medarde, Rogelio González-Sarmiento, Rafael Peláez

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Kinetic and structural studies on the interactions of Torpedo californica acetylcholinesterase with two donepezil-like rigid analogues by Rosanna Caliandro, Alessandro Pesaresi, Luca Cariati, Antonio Procopio, Manuela Oliverio, Doriano Lamba

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Identification of novel indole derivatives acting as inhibitors of the Keap1-Nrf2 interaction by Barbara Cosimelli, Giovanni Greco, Sonia Laneri, Ettore Novellino, Antonia Sacchi, Giorgio Amendola, Sandro Cosconati, Roberta Bortolozzi, Giampietro Viola

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Nimesulide linked acyl thioureas potent carbonic anhydrase I, II and α-glucosidase inhibitors: Design, synthesis and molecular docking studies by Atteeque Ahmed, Imran Shafique, Aamer Saeed, Ghulam Shabir, Arslan Saleem, Parham Taslimi, Tugba Taskin Tok, Mahinur Kirici, Eda Mehtap Üç, Muhammad Zaffar Hashmi

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The carbonic anhydrase IX inhibitor SLC-0111 sensitises cancer cells to conventional chemotherapy by Elena Andreucci, Jessica Ruzzolini, Silvia Peppicelli, Francesca Bianchini, Anna Laurenzana, Fabrizio Carta, Claudiu T. Supuran, Lido Calorini

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Synthesis, characterisation, biological evaluation and in silico studies of sulphonamide Schiff bases by Mustafa Durgun, Cüneyt Türkeş, Mesut Işık, Yeliz Demir, Ali Saklı, Ali Kuru, Abdussamat Güzel, Şükrü Beydemir, Suleyman Akocak, Sameh M. Osman, Zeid AlOthman, Claudiu T. Supuran

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Novel 1-(2-pyrimidin-2-yl)piperazine derivatives as selective monoamine oxidase (MAO)-A inhibitors by Betül Kaya, Leyla Yurttaş, Begüm Nurpelin Sağlik, Serkan Levent, Yusuf Özkay, Zafer Asim Kaplancikli

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