Search Results - "Medicinal Chemistry"

Quetiapine and novel PDE10A inhibitors potentiate the anti-BuChE activity of donepezil by Joanna Sikora, Maria Podsiedlik, Tadeusz Pietras, Marcin Kosmalski, Mikołaj Matłoka, Rafał Moszczyński-Petkowski, Maciej Wieczorek, Magdalena Markowicz-Piasecka

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Novel tacrine-benzofuran hybrids as potential multi-target drug candidates for the treatment of Alzheimer's Disease by Gaia Fancellu, Karam Chand, Daniel Tomás, Elisabetta Orlandini, Luca Piemontese, Diana F. Silva, Sandra M. Cardoso, Sílvia Chaves, M. Amélia Santos

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Novel sulfonamide benzoquinazolinones as dual EGFR/HER2 inhibitors, apoptosis inducers and radiosensitizers by Aiten M. Soliman, Ali S. Alqahtani, Mostafa M. Ghorab

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Novel N-Arylmethyl-aniline/chalcone hybrids as potential VEGFR inhibitors: synthesis, biological evaluations, and molecular dynamic simulations by Hesham Haffez, Nosaiba A. Elsayed, Marwa F. Ahmed, Samar S. Fatahala, Eman F. Khaleel, Rehab Mustafa Badi, Eslam B. Elkaeed, Mahmoud A. El Hassab, Sherif F. Hammad, Wagdy M. Eldehna, Nicolas Masurier, Radwan El-Haggar

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Hyperbaric oxygen therapy ameliorates osteonecrosis in patients by modulating inflammation and oxidative stress by Gerardo Bosco, Giuliano Vezzani, Simona Mrakic Sposta, Alex Rizzato, Garrett Enten, Abdullah Abou-samra, Sandro Malacrida, Silvia Quartesan, Alessandra Vezzoli, Enrico Camporesi

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New natural protein tyrosine phosphatase 1B inhibitors from Gynostemma pentaphyllum by Xianting Wang, Yidan Deng, Jianmei Wang, Lin Qin, Yimei Du, Qianru Zhang, Di Wu, Xingdong Wu, Jian Xie, Yuqi He, Daopeng Tan

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Comparison of blood carbonic anhydrase activity of athletes performing interval and continuous running exercise at high altitude by Murat Tas, Esra Senturk, Deniz Ekinci, Ramazan Demirdag, Veysal Comakli, Metin Bayram, Murat Akyuz, Murat Senturk, Claudiu T. Supuran

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Xanthones Active against Multidrug Resistance and Virulence Mechanisms of Bacteria by Fernando Durães, Diana I. S. P. Resende, Andreia Palmeira, Nikoletta Szemerédi, Madalena M. M. Pinto, Gabriella Spengler, Emília Sousa

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Design, synthesis and biological evaluation of novel histone deacetylase (HDAC) inhibitors derived from β-elemene scaffold by Yuan Gao, Jilong Duan, Xiawen Dang, Yinghui Yuan, Yu Wang, Xingrui He, Renren Bai, Xiang-Yang Ye, Tian Xie

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Discovery of cyanopyridine scaffold as novel indoleamine-2,3-dioxygenase 1 (IDO1) inhibitors through virtual screening and preliminary hit optimisation by Xi Xu, Jie Ren, Yinghe Ma, Hongting Liu, Quanjin Rong, Yifan Feng, Yameng Wang, Yu Cheng, Ruijia Ge, Zhiyu Li, Jinlei Bian

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Ultrasound promoted green synthesis, anticancer evaluation, and molecular docking studies of hydrazines: a pilot trial by Amena Ali, Abuzer Ali, Abu Tahir, Mohammed Afroz Bakht, Mohamed Jawed Ahsan

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Synthesis, biological evaluation, and molecular modelling studies of potent human neutrophil elastase (HNE) inhibitors by Maria Paola Giovannoni, Igor A. Schepetkin, Mark T. Quinn, Niccolò Cantini, Letizia Crocetti, Gabriella Guerrini, Antonella Iacovone, Paola Paoli, Patrizia Rossi, Gianluca Bartolucci, Marta Menicatti, Claudia Vergelli

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Organoboronic acids/esters as effective drug and prodrug candidates in cancer treatments: challenge and hope by Mothana K. Al-Omari, Mai Elaarag, Raed M. Al-Zoubi, Ahmad R. Al-Qudimat, Ayman A. Zarour, Enas A. Al-Hurani, Zainab E. Fares, Leena M. Alkharraz, Mohanad Shkoor, Abdulilah D. Bani-Yaseen, Omar M. Aboumarzouk, Aksam Yassin, Abdulla A. Al-Ansari

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Understanding the mechanism of ulcerative colitis-induced colorectal cancer and revealing the potential of Dillenia Indica in its management by Sujata Paul, El Bethel Lalthavel Hmar, Hemanta Kumar Sharma

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Identification of imidazo[4,5-c]pyridin-2-one derivatives as novel Src family kinase inhibitors against glioblastoma by Lishun Zhang, Zichao Yang, Huiting Sang, Ying Jiang, Mingfeng Zhou, Chuan Huang, Chunhui Huang, Xiaoyun Wu, Tingting Zhang, Xingmei Zhang, Shanhe Wan, Jiajie Zhang

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Novel Au Carbene Complexes as Promising Multi-Target Agents in Breast Cancer Treatment by Jessica Ceramella, Annaluisa Mariconda, Marco Sirignano, Domenico Iacopetta, Camillo Rosano, Alessia Catalano, Carmela Saturnino, Maria Stefania Sinicropi, Pasquale Longo

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Cover, Content, and Editorial Note from Borneo J Pharm Vol. 5 No. 4 November 2022 by Chief Editor of Borneo J Pharm

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Synthesis of new pyridothienopyrimidinone derivatives as Pim-1 inhibitors by Bassem H. Naguib, Hala B. El-Nassan, Tamer M. Abdelghany

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Cover, Content, and Editorial Note from Borneo J Pharm Vol. 6 No. 1 February 2023 by Chief Editor of Borneo J Pharm

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Cytotoxic substituted indolizines as new colchicine site tubulin polymerisation inhibitors by Monica-Cornelia Sardaru, Anda Mihaela Craciun, Cristina-Maria Al Matarneh, Isabela Andreea Sandu, Roxana Maria Amarandi, Lacramioara Popovici, Catalina Ionica Ciobanu, Dragos Peptanariu, Mariana Pinteala, Ionel I. Mangalagiu, Ramona Danac

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