Search Results - "structure–activity relationship"

Synthesis and anаlgеsic activity 5-methyl-3-aryl[1,2,4]triazolo[4,3-a]pyrimidin-7-oles derivatives by A. G. Ogorodnik, V. A. Yanchenko, L. S. Bobkova, N. M. Seredinska, A. M. Demchenko

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Design, synthesis, in vitro antiproliferative activity and apoptosis-inducing studies of 1-(3',4',5'-trimethoxyphenyl)-3-(2'-alkoxycarbonylindolyl)-2-propen-1-one derivatives obtai... by Delia Preti, Romeo Romagnoli, Riccardo Rondanin, Barbara Cacciari, Ernest Hamel, Jan Balzarini, Sandra Liekens, Dominique Schols, Francisco Estévez-Sarmiento, José Quintana, Francisco Estévez

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Using drug chemical structures in the education of pharmacology and clinical therapeutics key concepts by Ghina'a Ismail Abu Deiab, Loai Mohammed Saadah, Iman Amin Basheti

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Search for structurally diverse heterocyclic analogs as dual-acting antimalarial and antileishmanial agents: An overview by Faheem, Sanchita Dey, Samridhi Johri, M. Abirami, Banoth Karan Kumar, Donatella Taramelli, Nicoletta Basilico, Rafael Balana-Fouce, Kondapalli Venkata Gowri Chandra Sekhar, Sankaranarayanan Murugesan

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Cytotoxicity of some 1-(2,4-dihydroxyphenyl)-3-(4-phenylpiperidin-1-yl) prop-2-en-1-one derivatives using MTT assay by Farzaneh Fesahat, Mehdi Khoshneviszadeh, Alireza Foroumadi, Alireza Vahidi, Maryam Fereidounpour, Amirhossein Sakhteman

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Bioisosteric modification on melatonin: synthesis of new naphthalene derivatives, in vitro antioxidant activity and cytotoxicity studies by Hanif Shirinzadeh, Mohammed Ghalia, Alev Tascioglu, Ferial Intissar Adjali, Gulsen Gunesacar, Hande Gurer-Orhan, Sibel Suzen

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Cytotoxicity of some 1-(2,4-dihydroxyphenyl)-3-(4-phenylpiperidin-1-yl) prop-2-en-1-one derivatives using MTT assay by Farzaneh Fesahat, Mehdi Khoshneviszadeh, Alireza Foroumadi, Alireza Vahidi, Maryam Fereidounpour, Amirhossein Sakhteman

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Lipid Membranes as Key Targets for the Pharmacological Actions of Ginsenosides by Sandrine L. Verstraeten, Joseph H. Lorent, Joseph H. Lorent, Marie-Paule M

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CoMFA and docking study of 2,N6-disubstituted 1,2-dihydro-1,3,5-triazine-4,6-diamines as novel PfDHFR enzyme inhibitors for antimalarial activity by Pritam N. Dube, Santosh Mokale, Prasanna Datar

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Synthesis and biological evaluation of sophocarpinic acid derivatives as anti-HCV agents by Yinghong Li, Zonggen Peng, Limei Gao, Danqing Song

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Medicinal Chemistry of Quinazolines as Anticancer Agents Targeting Tyrosine Kinases by Mohamed F. Zayed

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A Pharmacological Overview of Alpinumisoflavone, a Natural Prenylated Isoflavonoid by Sylvin Benjamin Ateba, Marie Alfrede Mvondo, Sefirin Djiogue, Stéphane Zingué, Liselotte Krenn, Dieudonné Njamen

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Synthetic Imidazopyridine-Based Derivatives as Potential Inhibitors against Multi-Drug Resistant Bacterial Infections: A Review by Bharat Kumar Reddy Sanapalli, Akram Ashames, Dilep Kumar Sigalapalli, Afzal B. Shaik, Richie R. Bhandare, Vidyasrilekha Yele

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Benzimidazole and its derivatives as cancer therapeutics: The potential role from traditional to precision medicine by Yeuan Ting Lee, Yi Jer Tan, Chern Ein Oon

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Synthesis, biological and computational evaluation of novel cyanomethyl vinyl ether derivatives by Endika Martín-Encinas, María Fuertes, Samuel Delgado-Hernández, Fernando García-Tellado, David Tejedor, Concepción Alonso

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Tetrahydroquinazole-based secondary sulphonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IV, and IX, and computational studies by Emma Baglini, Rahul Ravichandran, Emanuela Berrino, Silvia Salerno, Elisabetta Barresi, Anna Maria Marini, Monica Viviano, Sabrina Castellano, Federico Da Settimo, Claudiu T. Supuran, Sandro Cosconati, Sabrina Taliani

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Recent Research Advances in Small-Molecule Pan-PIM Inhibitors by Lei Xu, Yu-Cheng Meng, Peng Guo, Ming Li, Lei Shao, Jun-Hai Huang

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Structural diversity and biological activities of caged Garcinia xanthones: recent updates by Yee Lin Phang, Changwu Zheng, Hongxi Xu

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Structural/Functional Matches and Divergences of Phytoprostanes and Phytofurans with Bioactive Human Oxylipins by Sonia Medina, Ángel Gil-Izquierdo, Thierry Durand, Federico Ferreres, Raúl Domínguez-Perles

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Synthesis and biological evaluation of 8-substituted berberine derivatives as novel anti-mycobacterial agents by Yanxiang Wang, Haigen Fu, Yinghong Li, Jiandong Jiang, Danqing Song

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