Search Results - "structure–activity relationship"

Aryl derivatives of 3H-1,2-benzoxaphosphepine 2-oxides as inhibitors of cancer-related carbonic anhydrase isoforms IX and XII by Anastasija Balašova, Aleksandrs Pustenko, Alessio Nocentini, Daniela Vullo, Claudiu T. Supuran, Raivis Žalubovskis

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Phenolic Compounds in Bacterial Inactivation: A Perspective from Brazil by Angélica Correa Kauffmann, Vinicius Silva Castro

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The Role of Five-Membered Heterocycles in the Molecular Structure of Antibacterial Drugs Used in Therapy by Aura Rusu, Ioana-Maria Moga, Livia Uncu, Gabriel Hancu

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Sinapic Acid Esters: Octinoxate Substitutes Combining Suitable UV Protection and Antioxidant Activity by Cédric Peyrot, Matthieu M. Mention, Fanny Brunissen, Florent Allais

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Biosynthesis and Chemical Synthesis of Albomycin Nucleoside Antibiotics by Meiyan Wang, Yuxin Zhang, Lanxin Lv, Dekun Kong, Guoqing Niu

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Pyrazole and Triazole Derivatives as <i>Mycobacterium tuberculosis</i> UDP-Galactopyranose Inhibitors by Dalia M. Ahmed, Jeffrey M. Chen, David A. R. Sanders

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Synthesis of Alkyne-Substituted Dihydropyrrolones as Bacterial Quorum-Sensing Inhibitors of <i>Pseudomonas aeruginosa</i> by Basmah Almohaywi, Tsz Tin Yu, George Iskander, Shekh Sabir, Mohan Bhadbhade, David StC. Black, Naresh Kumar

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New Insights on the Mechanism of Fatty Acids as Buccal Permeation Enhancers by Cristina Padula, Silvia Pescina, Sara Nicoli, Patrizia Santi

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Pharmacophore-based discovery of 2-(phenylamino)aceto-hydrazides as potent eosinophil peroxidase (EPO) inhibitors by Daniela Schuster, Martina Zederbauer, Thierry Langer, Andreas Kubin, Paul G. Furtmüller

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Antibody-drug conjugates: Recent advances in payloads by Zhijia Wang, Hanxuan Li, Lantu Gou, Wei Li, Yuxi Wang

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Extensive expansion of the chemical diversity of fusidane-type antibiotics using a stochastic combinational strategy by Xiaojun Song, Jianming Lv, Zhiqin Cao, Huiyun Huang, Guodong Chen, Takayoshi Awakawa, Dan Hu, Hao Gao, Ikuro Abe, Xinsheng Yao

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Molecular Determinants Responsible for Sedative and Non-sedative Properties of Histamine H1-Receptor Antagonists by Yoshihiro Uesawa, Shigeru Hishinuma, Masaru Shoji

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Rational drug design, synthesis, and biological evaluation of novel chiral tetrahydronaphthalene-fused spirooxindole as MDM2-CDK4 dual inhibitor against glioblastoma by Biao Wang, Fu Peng, Wei Huang, Jin Zhou, Nan Zhang, Jia Sheng, Phensinee Haruehanroengra, Gu He, Bo Han

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Upregulation of p53 through induction of MDM2 degradation: improved potency through the introduction of an alkylketone sidechain on the anthraquinone core by Ravi Tripathi, Abiodun Anifowose, Wen Lu, Xiaoxiao Yang, Binghe Wang

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Development of QSAR models to predict blood-brain barrier permeability by Sadegh Faramarzi, Marlene T. Kim, Donna A. Volpe, Kevin P. Cross, Suman Chakravarti, Lidiya Stavitskaya

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Technologies for Direct Detection of Covalent Protein-Drug Adducts by Elma Mons, Robbert Q. Kim, Monique P. C. Mulder

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Discovery and development of Factor Xa inhibitors (2015-2022) by Wei Zheng, Wei Zheng, Xiaoqin Dai, Binyao Xu, Wei Tian, Jianyou Shi

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Isatin Bis-Imidathiazole Hybrids Identified as FtsZ Inhibitors with On-Target Activity Against <i>Staphylococcus aureus</i> by Rita Morigi, Daniele Esposito, Matteo Calvaresi, Tainah Dorina Marforio, Giovanna Angela Gentilomi, Francesca Bonvicini, Alessandra Locatelli

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Hydrazone-Containing Triblock Copolymeric Micelles for pH-Controlled Drug Delivery by Peilan Qi, Xiaohe Wu, Lei Liu, Huimin Yu, Shiyong Song

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A Review of Antioxidant Peptides Derived from Meat Muscle and By-Products by Rui Liu, Lujuan Xing, Qingquan Fu, Guang-hong Zhou, Wan-gang Zhang

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