Search Results - "structure–activity relationship"

QSAR BERBASIS DESKRIPTOR GRAF DAN MOLECULAR DOCKING DARI TURUNAN FENILPIRIMIDIN SEBAGAI ANTIJAMUR S. SCLEROTIORUM by Tria Nurwina Novianti, -

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SCREENING ANTIDOT OKSIM NON-KUARTERNER DAN NON-OKSIM SEBAGAI REAKTIVATOR ASETILKOLINESTERASE TERINHIBISI ORGANOFOSFAT DENGAN 3D-QSAR DAN MOLECULAR DOCKING by Zachnaz Fairuuz, -

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Physiology and Pathophysiology of Proteinase-Activated Receptors (PARs): PAR-2 as a Potential Therapeutic Target by Toru Kanke, Toshiaki Takizawa, Mototsugu Kabeya, Atsufumi Kawabata

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A comprehensive review on pyrazoline based heterocyclic hybrids as potent anticancer agents by Kashif Haider, Mohd Shafeeque, Shaikh Yahya, M. Shahar Yar

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Synthesis of hydrazides of heterocyclic amines and their antimicrobial and spasmolytic activity by Dmitriy A. Berillo, Moldyr A. Dyusebaeva

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The future of pharmacology and therapeutics of the arachidonic acid cascade in the next decade: Innovative advancements in drug repurposing by Paola Patrignani, Paola Patrignani, Annalisa Contursi, Annalisa Contursi, Stefania Tacconelli, Stefania Tacconelli, Dieter Steinhilber

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The hop-derived compounds xanthohumol, isoxanthohumol and 8-prenylnaringenin are tight-binding inhibitors of human aldo-keto reductases 1B1 and 1B10 by Jan Moritz Seliger, Livia Misuri, Edmund Maser, Jan Hintzpeter

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The Antimicrobial Peptide Capitellacin: Chemical Synthesis of Analogues to Probe the Role of Disulphide Bridges and Their Replacement with Vinyl Sulphides by Oscar A. Shepperson, Paul W. R. Harris, Margaret A. Brimble, Alan J. Cameron

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Discovery of Ureido-Based Apcin Analogues as Cdc20-specific Inhibitors against Cancer by Yiqin He, Xiangyang Le, Gaoyun Hu, Qianbin Li, Zhuo Chen

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4-Anilinoquinazoline-based benzenesulfonamides as nanomolar inhibitors of carbonic anhydrase isoforms I, II, IX, and XII: design, synthesis, in-vitro, and in-silico biological stud... by Hossam Nada, Ahmed Elkamhawy, Magda H. Abdellattif, Andrea Angeli, Chang Hoon Lee, Claudiu T. Supuran, Kyeong Lee

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Synthesis and bioevaluation of new tacrine-cinnamic acid hybrids as cholinesterase inhibitors against Alzheimer's disease by Yao Chen, Jie Zhu, Jun Mo, Hongyu Yang, Xueyang Jiang, Hongzhi Lin, Kai Gu, Yuqiong Pei, Liang Wu, Renxiang Tan, Jing Hou, Jingyi Chen, Yang Lv, Yaoyao Bian, Haopeng Sun

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Design and synthesis of doublecortin-like kinase 1 inhibitors and their bioactivity evaluation by Pengming Pan, Dengbo Ji, Zhongjun Li, Xiangbao Meng

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Dimethyl Itaconate Inhibits Melanogenesis in B16F10 Cells by Bo-Yeong Yu, Hoang Hai Ngo, Won Jun Choi, Young-Sam Keum

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Synthesis, in vitro inhibitory activity, kinetic study and molecular docking of novel N-alkyl-deoxynojirimycin derivatives as potential α-glucosidase inhibitors by Ping Lin, Jia-Cheng Zeng, Ji-Guang Chen, Xu-Liang Nie, En Yuan, Xiao-Qiang Wang, Da-Yong Peng, Zhong-Ping Yin

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Evaluation of Heterocyclic Carboxamides as Potential Efflux Pump Inhibitors in <i>Pseudomonas aeruginosa</i> by Yi Yuan, Jesus D. Rosado-Lugo, Yongzheng Zhang, Pratik Datta, Yangsheng Sun, Yanlu Cao, Anamika Banerjee, Ajit K. Parhi

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Identification of Novel Chemical Scaffolds that Inhibit the Growth of Mycobacterium tuberculosis in Macrophages by Sara Ahmed, Sara Ahmed, Alyssa Manning, Lindsay Flint, Divya Awasthi, Yulia Ovechkina, Tanya Parish, Tanya Parish

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A Concise Review of the Recent Structural Explorations of Chromones as MAO-B Inhibitors: Update from 2017 to 2023 by Reshma Susan Ipe, Sunil Kumar, Feba Benny, Jayalakshmi Jayan, Amritha Manoharan, Sachitra Thazhathuveedu Sudevan, Ginson George, Prashant Gahtori, Hoon Kim, Bijo Mathew

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Identification of Mepenzolate Derivatives With Long-Acting Bronchodilatory Activity by Ken-Ichiro Tanaka, Naoki Yamakawa, Yasunobu Yamashita, Teita Asano, Yuki Kanda, Ayaka Takafuji, Masahiro Kawahara, Mitsuko Takenaga, Yoshifumi Fukunishi, Tohru Mizushima

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C-2 phenyl replacements to obtain potent quinoline-based Staphylococcus aureus NorA inhibitors by Tommaso Felicetti, Gianmarco Mangiaterra, Rolando Cannalire, Nicholas Cedraro, Donatella Pietrella, Andrea Astolfi, Serena Massari, Oriana Tabarrini, Giuseppe Manfroni, Maria Letizia Barreca, Violetta Cecchetti, Francesca Biavasco, Stefano Sabatini

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Phenols and GABAA receptors: from structure and molecular mechanisms action to neuropsychiatric sequelae by Sergey A. Menzikov, Danila M. Zaichenko, Aleksey A. Moskovtsev, Sergey G. Morozov, Aslan A. Kubatiev

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