Search Results - "structure–activity relationship"

In vitro antimicrobial combat, molecular modelling and structure activity relationship studies of novel class of aryl-ethyne tethered coumarin analogues and some 3-aryl coumarin derivatives by Pavankumar Prabhala, Suraj M. Sutar, Hemantkumar M. Savanur, Shrinivas D. Joshi, Rajesh G. Kalkhambkar

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Synthesis, docking study, and structure activity relationship of novel anti-tumor 1, 2, 4 triazole derivatives incorporating 2-(2, 3- dimethyl aminobenzoic acid) moiety by Hiba Alsaad, Ammar Kubba, Lubna H. Tahtamouni, Ali H. Hamzah

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Structure-Activity Relationship Studies of 9-Alkylamino-1,2,3,4-tetrahydroacridines against <i>Leishmania</i> (<i>Leishmania</i>) <i>infantum</i> Promastigotes by Carlos F. M. Silva, Teresa Leão, Filipa Dias, Ana M. Tomás, Diana C. G. A. Pinto, Eduardo F. T. Oliveira, Ana Oliveira, Pedro A. Fernandes, Artur M. S. Silva

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Design, synthesis and structure-activity relationship studies of 3-phenylpyrazino[1,2-a]indol-1(2H)-ones as amyloid aggregation and cholinesterase inhibitors with antioxidant activity by Sarbjeet Singh Gujral, Arash Shakeri, Leila Hejazi, Praveen P.N. Rao

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Discovery of a series of dimethoxybenzene FGFR inhibitors with 5H-pyrrolo[2,3-b]pyrazine scaffold: structure-activity relationship, crystal structural characterization and in vivo study by Peng Wei, Bo Liu, Ruifeng Wang, Yinglei Gao, Lanlan Li, Yuchi Ma, Zhiwei Qian, Yuelei Chen, Maosheng Cheng, Meiyu Geng, Jingkang Shen, Dongmei Zhao, Jing Ai, Bing Xiong

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Kassporin-KS1: A Novel Pentadecapeptide from the Skin Secretion of <i>Kassina senegalensis</i>: Studies on the Structure-Activity Relationships of Site-Specific "Glycine-Lysine" Motif Insertions by Yueyang Lu, Wanchen Zou, Lei Wang, Xinping Xi, Chengbang Ma, Xiaoling Chen, Tianbao Chen, Chris Shaw, Xu Zhang, Mei Zhou

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Investigation into the Interaction between Penicillin-Resistant and Penicillin-Susceptible Gonococcal Penicillin-Binding Protein 2 and Target Phenolic Ligands through Molecular Docking Studies and Structure-Activity Relationship Analysis by Sinethemba Yakobi, Lindiwe Zuma, Ofentse Pooe

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Structure-Activity Relationship of Synthetic Linear KTS-Peptides Containing Meta-Aminobenzoic Acid as Antagonists of α1β1 Integrin with Anti-Angiogenic and Melanoma Anti-Tumor Activities by Majdi Saleem Naamneh, Tatjana Momic, Michal Klazas, Julius Grosche, Johannes A. Eble, Cezary Marcinkiewicz, Netaly Khazanov, Hanoch Senderowitz, Amnon Hoffman, Chaim Gilon, Jehoshua Katzhendler, Philip Lazarovici

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New horizons in drug discovery of lymphocyte-specific protein tyrosine kinase (Lck) inhibitors: a decade review (2011-2021) focussing on structure-activity relationship (SAR) and docking insights by Ahmed Elkamhawy, Eslam M. H. Ali, Kyeong Lee

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The Molecular Aspect of Natural Secondary Metabolite Products in Health and Disease by Toshio Morikawa (Ed.)

Subjects: “…structure-activity relationship…”
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Design and Synthesis of Novel 5-((3-(Trifluoromethyl)piperidin-1-yl)sulfonyl)indoline-2,3-dione Derivatives as Promising Antiviral Agents: In Vitro, In Silico, and Structure-Activity Relationship Studies by Rogy R. Ezz Eldin, Marwa A. Saleh, Sefat A. Alwarsh, Areej Rushdi, Azza Ali Althoqapy, Hoda S. El Saeed, Ayman Abo Elmaaty

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Effects of Synthetic Sphingosine-1-Phosphate Analogs on Cytosolic Phospholipase A2α-Independent Release of Arachidonic Acid and Cell Toxicity in L929 Fibrosarcoma Cells: the Structure-Activity Relationship by Masaya Shimizu, Yuki Muramatsu, Eiko Tada, Takeshi Kurosawa, Erika Yamaura, Hiroyuki Nakamura, Hiromichi Fujino, Yuuya Houjyo, Yuri Miyasaka, Yuuki Koide, Atsushi Nishida, Toshihiko Murayama

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Synthesis and Structure-Activity Relationships for the Anti-Mycobacterial Activity of 3-Phenyl-<i>N</i>-(Pyridin-2-ylmethyl)Pyrazolo[1,5-<i>a</i>]Pyrimidin-7-Amines by Hamish S. Sutherland, Peter J. Choi, Guo-Liang Lu, Anna C. Giddens, Amy S. T. Tong, Scott G. Franzblau, Christopher B. Cooper, Brian D. Palmer, William A. Denny

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Synthesis and preliminary structure-activity relationship study of 2-aryl-2H-pyrazolo[4,3-c]quinolin-3-ones as potential checkpoint kinase 1 (Chk1) inhibitors by Ivana Malvacio, Alberto Cuzzolin, Mattia Sturlese, D. Mariano A. Vera, E. Laura Moyano, Stefano Moro

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USING QUANTUM-CHEMICAL PARAMETERS FOR PREDICTING ANTIRADICAL (HO•) ACTIVITY OF RELATED STRUCTURES CONTAINING A CINNAMOIL FRAGMENT. IV. STRUCTURE-ACTIVITY RELATIONSHIP BETWEEN UNSATURATION INDICES AND FLAVONE DERIVATIVES WITH FLOROGLUCIN RING "A" by E. T. Oganesyan, S. S. Shatokhin

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Biological Activity of Natural Secondary Metabolite Products by Toshio Morikawa (Ed.)

Subjects: “…structure-activity relationship…”
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Natural Products from Marine Microorganisms

Subjects: “…structure-activity relationships…”
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Screening of anxiolytic properties and analysis of structure-activity relationship of new derivatives of 6-(4-methoxy)-7H-[1,2,4]triazolo[3,4-a][2,3]benzodiazepine under the code RD by Maria O. Skripka, Alexander A. Spasov, Dmitriy V. Maltsev, Mikhail V. Miroshnikov, Dmitriy S. Yakovlev, Kira T. Sultanova, Maxim A. Kochergin, Lyudmila N. Divaeva

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Synthesis and Regularities of the Structure-Activity Relationship in a Series of <i>N</i>-Pyridyl-4-methyl-2,2-dioxo-1<i>H</i>-2λ⁶,1-benzothiazine-3-carboxamides by Igor V. Ukrainets, Anna A. Burian, Ganna M. Hamza, Natali I. Voloshchuk, Oxana V. Malchenko, Svitlana V. Shishkina, Lyudmila V. Sidorenko, Kateryna O. Burian, Galina Sim

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Structure-Activity Relationship of <i>N</i>-Phenylthieno[2,3-<i>b</i>]pyridine-2-carboxamide Derivatives Designed as Forkhead Box M1 Inhibitors: The Effect of Electron-Withdrawing and Donating Substituents on the Phenyl Ring by César Sebastian Huerta-García, David J. Pérez, Carlos A. Velázquez-Martínez, Seyed Amirhossein Tabatabaei Dakhili, Antonio Romo-Mancillas, Rafael Castillo, Alicia Hernández-Campos

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