Subcellular localization of several structurally different tyrosine kinase inhibitors

Protein tyrosine kinases form an important target for a new class of anticancer drugs, the tyrosine kinase inhibitors (TKIs). Recently we demonstrated that sunitinib, an inhibitor of the membrane-associated vascular endothelial growth factor receptor (VEGFR), is trapped in lysosomes which isolates t...

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Egile Nagusiak: Richard Honeywell (Egilea), Sarina Hitzerd (Egilea), Ietje Kathmann (Egilea), Godefridus Peters (Egilea)
Formatua: Liburua
Argitaratua: International Association of Physical Chemists (IAPC), 2018-09-01T00:00:00Z.
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