New potent steroid sulphatase inhibitors based on 6-(1-phenyl-1H-1,2,3-triazol-4-yl)naphthalen-2-yl sulphamate derivatives

In the present work, we report a new class of potent steroid sulphatase (STS) inhibitors based on 6-(1-phenyl-1H-1,2,3-triazol-4-yl)naphthalen-2-yl sulphamate derivatives. Within the set of new STS inhibitors, 6-(1-(1,2,3-trifluorophenyl)-1H-1,2,3-triazol-4-yl)naphthalen-2-yl sulphamate 3L demonstra...

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Main Authors: Olga Ciupak (Author), Mateusz Daśko (Author), Karol Biernacki (Author), Janusz Rachon (Author), Maciej Masłyk (Author), Konrad Kubiński (Author), Aleksandra Martyna (Author), Sebastian Demkowicz (Author)
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Publicado em: Taylor & Francis Group, 2021-01-01T00:00:00Z.
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