Strategies to overcome drug resistance using SHP2 inhibitors
Encoded by PTPN11, the SHP2 (Src homology-2 domain-containing protein tyrosine phosphatase-2) is widely recognized as a carcinogenic phosphatase. As a promising anti-cancer drug target, SHP2 regulates many signaling pathways such as RAS-RAF-ERK, PI3K-AKT and JAK-STAT. Meanwhile, SHP2 plays a signifi...
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Materiálatiipa: | Girji |
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Elsevier,
2021-12-01T00:00:00Z.
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