Synthesis and biological assessment of indole derivatives containing penta-heterocycles scaffold as novel anticancer agents towards A549 and K562 cells

Herein, a new series of 2-chloro-N-(5-(2-oxoindolin-3-yl)-4H-pyrazol-3-yl) acetamide derivatives containing 1,3,4-thiadiazole (10a-i) and 4H-1,2,4-triazol-4-amine (11a-r) moiety was designed, synthesised as novel anticancer agents. The antiproliferative activity values indicated that compound 10 b s...

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Váldodahkkit: Guanglong Zhang (Dahkki), Zhenhua Tang (Dahkki), Sili Fan (Dahkki), Chengpeng Li (Dahkki), Yan Li (Dahkki), Weiqin Liu (Dahkki), Xuesha Long (Dahkki), Wenjing Zhang (Dahkki), Yi Zhang (Dahkki), Zhurui Li (Dahkki), Zhenchao Wang (Dahkki), Danping Chen (Dahkki), Guiping Ouyang (Dahkki)
Materiálatiipa: Girji
Almmustuhtton: Taylor & Francis Group, 2023-12-01T00:00:00Z.
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3rd Floor Main Library

oažžasuvvan: 3rd Floor Main Library
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