Novel inhibitors of phosphorylation independent activity of GRK2 modulate cAMP signaling
Abstract G protein‐coupled receptors kinase 2 (GRK2) plays a major role in receptor regulation and, as a consequence, in cell biology and physiology. GRK2‐mediated receptor desensitization is performed by its kinase domain, which exerts receptor phosphorylation promoting G protein uncoupling and the...
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Main Authors: | Emiliana Echeverría (Author), Sonia Ripoll (Author), Lucas Fabián (Author), Carina Shayo (Author), Federico Monczor (Author), Natalia C. Fernández (Author) |
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Format: | Book |
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Wiley,
2022-04-01T00:00:00Z.
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Online Access: | Connect to this object online. |
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