Evaluation of Actinium-225 Labeled Minigastrin Analogue [<sup>225</sup>Ac]Ac-DOTA-PP-F11N for Targeted Alpha Particle Therapy

The overexpression of cholecystokinin B receptor (CCKBR) in human cancers led to the development of radiolabeled minigastrin analogues for targeted radionuclide therapy, which aims to deliver cytotoxic radiation specifically to cancer cells. Alpha emitters (e.g., actinium-225) possess high potency i...

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Egile Nagusiak: Yun Qin (Egilea), Stefan Imobersteg (Egilea), Alain Blanc (Egilea), Stephan Frank (Egilea), Roger Schibli (Egilea), Martin P. Béhé (Egilea), Michal Grzmil (Egilea)
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Argitaratua: MDPI AG, 2020-11-01T00:00:00Z.
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