Co-Amorphous Solid Dispersion System for Improvement in Dissolution Profile of <i>N</i>-(((1<i>r</i>,4<i>r</i>)-4-((6-fluorobenzo[<i>d</i>]oxazol-2-yl)amino)cyclohexyl)methyl)-2-methylpropane-2-sulfonamide as a Neuropeptide Y5 Receptor Antagonist

<b>Background/Objectives:</b> Brick dust molecules exhibit high melting points and ultralow solubility. Overcoming this solubility issue is challenging. Previously, we formulated a co-amorphous system for a neuropeptide Y5 receptor antagonist (NP) as a brick dust drug using sodium tauroc...

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Autores principales: Hironori Tanaka (Autor), Hiroshi Ueda (Autor)
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Publicado: MDPI AG, 2024-10-01T00:00:00Z.
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