Styrylquinazoline derivatives as ABL inhibitors selective for different DFG orientations

Among tyrosine kinase inhibitors, quinazoline-based compounds represent a large and well-known group of multi-target agents. Our previous studies have shown interesting kinases inhibition activity for a series of 4-aminostyrylquinazolines based on the CP-31398 scaffold. Here, we synthesised a new se...

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Autores principales: Katarzyna Malarz (Autor), Jacek Mularski (Autor), Marcin Pacholczyk (Autor), Robert Musiol (Autor)
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Publicado: Taylor & Francis Group, 2023-12-01T00:00:00Z.
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