Covalent modification of nephrilin peptide with valproic acid increases its efficacy as a therapeutic in burn trauma

Introduction: Nephrilin peptide, a designed inhibitor of Rictor complex, modulates systemic responses to trauma, alleviating clinically relevant variables in a rat scald model and sepsis mortality in a mouse model. This study explores the possibility that chemical conjugation of small molecules to t...

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Autores principales: Desmond D. Mascarenhas (Autor), Puja Ravikumar (Autor), Edward P. Amento (Autor)
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Publicado: Elsevier, 2020-07-01T00:00:00Z.
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