Multipotent cholinesterase/monoamine oxidase inhibitors for the treatment of Alzheimer’s disease: design, synthesis, biochemical evaluation, ADMET, molecular modeling, and QSAR analysis of novel donepezil-pyridyl hybrids

Oscar M Bautista-Aguilera,1,* Gerard Esteban,2,* Mourad Chioua,1 Katarina Nikolic,3 Danica Agbaba,3 Ignacio Moraleda,4 Isabel Iriepa,4 Elena Soriano,5 Abdelouahid Samadi,1 Mercedes Unzeta,2 José Marco-Contelles1 1Laboratory of Medicinal Chemistry (Institute of General Organic Chemistry [I...

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Main Authors: Bautista-Aguilera OM (Author), Esteban G (Author), Chioua M (Author), Nikolic K (Author), Agbaba D (Author), Moraleda I (Author), Iriepa I (Author), Soriano E (Author), Samadi A (Author), Unzeta M (Author), Marco-Contelles J (Author)
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Publicado em: Dove Medical Press, 2014-10-01T00:00:00Z.
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