α1-adrenoceptor ligands inhibit chemokine receptor heteromerization partners of α1B/D-adrenoceptors via interference with heteromer formation
We reported previously that α1-adrenoceptor (α1-AR) ligands inhibit chemokine receptor (CR) heteromerization partners of α1B/D-AR. The underlying mechanisms are unknown and in vivo evidence for such effects is missing. Utilizing CCR2 and α1B-AR as prototypical partners, we observed in recombinant sy...
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Main Authors: | Xianlong Gao (Author), Garrett A. Enten (Author), Michelle Y. McGee (Author), McWayne Weche (Author), Matthias Majetschak (Author) |
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Format: | Book |
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Elsevier,
2023-04-01T00:00:00Z.
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