GRPR-Antagonists Carrying DOTAGA-Chelator via Positively Charged Linkers: Perspectives for Prostate Cancer Theranostics

• Main Authors: Karim Obeid (Author), Panagiotis Kanellopoulos (Author), Ayman Abouzayed (Author), Adam Mattsson (Author), Vladimir Tolmachev (Author), Berthold A. Nock (Author), Theodosia Maina (Author), Anna Orlova (Author)
• Format: Book
• Published: MDPI AG, 2024-04-01T00:00:00Z.
• Subjects: article
• Online Access: Connect to this object online.

Gastrin-releasing peptide receptor (GRPR)-antagonists have served as motifs in the development of theranostic radioligands for prostate cancer. Our efforts have been focused on the development of radiolabeled RM26 (H-DPhe⁶-Gln⁷-Trp⁸...