Anti-breast cancer action of carbonic anhydrase IX inhibitor 4-[4-(4-Benzo[1,3]dioxol-5-ylmethyl-piperazin-1-yl)-benzylidene-hydrazinocarbonyl]-benzenesulfonamide (BSM-0004): in vitro and in vivo studies

Anti-breast cancer action of novel human carbonic anhydrase IX (hCA IX) inhibitor BSM-0004 has been investigated using in vitro and in vivo models of breast cancer. BSM-0004 was found to be a potent and selective hCA IX inhibitor with a Ki value of 96 nM. In vitro anticancer effect of BSM-0004 was a...

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Egile Nagusiak: Chandra Bhushan Mishra (Egilea), Raj Kumar Mongre (Egilea), Amresh Prakash (Egilea), Raok Jeon (Egilea), Claudiu T. Supuran (Egilea), Myeong-Sok Lee (Egilea)
Formatua: Liburua
Argitaratua: Taylor & Francis Group, 2021-01-01T00:00:00Z.
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