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Synthesis and Biological Evaluation of Indole-2-Carboxamides with Potent Apoptotic Antiproliferative Activity as EGFR/CDK2 Dual Inhibitors

The apoptotic antiproliferative actions of our previously reported CB1 allosteric modulators 5-chlorobenzofuran-2-carboxamide derivatives <b>VIIa</b>-<b>j</b> prompted us to develop and synthesise a novel series of indole-2-carboxamide derivatives <b>5a</b>-<b&...

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Main Authors:	Lamya H. Al-Wahaibi (Author), Yaser A. Mostafa (Author), Mostafa H. Abdelrahman (Author), Ali H. El-Bahrawy (Author), Laurent Trembleau (Author), Bahaa G. M. Youssif (Author)
Format:	Book
Published:	MDPI AG, 2022-08-01T00:00:00Z.
Subjects:	article
Online Access:	Connect to this object online.
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