Anticancer activity and toxicity of new quaternary ammonium geldanamycin derivative salts and their mixtures with potentiators

Geldanamycin (GDM) has been modified by different type neutral/acidic/basic substituents (1-7) and by quinuclidine motif (8), transformed into ammonium salts (9-13) at C(17). These compounds have been characterised by spectroscopic and x-ray methods. Derivative 8 shows better potency than GDM in MCF...

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Detaylı Bibliyografya
Asıl Yazarlar: Natalia Skrzypczak (Yazar), Krystian Pyta (Yazar), Piotr Ruszkowski (Yazar), Przemysław Mikołajczak (Yazar), Małgorzata Kucińska (Yazar), Marek Murias (Yazar), Maria Gdaniec (Yazar), Franz Bartl (Yazar), Piotr Przybylski (Yazar)
Materyal Türü: Kitap
Baskı/Yayın Bilgisi: Taylor & Francis Group, 2021-01-01T00:00:00Z.
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3rd Floor Main Library

Detaylı Erişim Bilgileri 3rd Floor Main Library
Yer Numarası: A1234.567
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