1-Oxo-3,4-dihydroisoquinoline-4-carboxamides as novel druglike inhibitors of poly(ADP-ribose) polymerase (PARP) with favourable ADME characteristics
A novel 3,4-dihydroisoquinol-1-one-4-carboxamide scaffold was designed as the basis for the development of novel inhibitors of poly(ADP-ribose) polymerase (PARP). Synthesis of 3,4-dihydroisoquinol-1-one-4-carboxylic acids was achieved using the previously developed protocol based on the modified Cas...
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Автори: | , , , , , , , |
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Формат: | Книга |
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Taylor & Francis Group,
2021-01-01T00:00:00Z.
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Connect to this object online.3rd Floor Main Library
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A1234.567 |
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Примірник 1 | Доступно |