Class I phosphatidylinositol 3-kinase inhibitors for cancer therapy

The phosphatidylinositol 3-kinase (PI3K) pathway is frequently activated in human cancers. Class I PI3Ks are lipid kinases that phosphorylate phosphatidylinositol 4,5-bisphosphate (PIP2) at the 3-OH of the inositol ring to generate phosphatidylinositol 3,4,5-trisphosphate (PIP3), which in turn activ...

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Main Authors: Wennan Zhao (Author), Yuling Qiu (Author), Dexin Kong (Author)
Formato: Livro
Publicado em: Elsevier, 2017-01-01T00:00:00Z.
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