Correlation of functional and radioligand binding characteristics of GPER ligands confirming aldosterone as a GPER agonist
Abstract Aldosterone exerts some of its effects not by binding to mineralocorticoid receptors, but rather by acting via G protein‐coupled estrogen receptors (GPER). To determine if aldosterone binds directly to GPER, we studied the ability of aldosterone to compete for the binding of [3H] 2‐methoxye...
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Main Authors: | Qingming Ding (Author), Jozef Chorazyczewski (Author), Robert Gros (Author), Harvey J. Motulsky (Author), Lee E. Limbird (Author), Ross D. Feldman (Author) |
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Format: | Book |
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Wiley,
2022-10-01T00:00:00Z.
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Online Access: | Connect to this object online. |
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