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Design and synthesis of some substituted thiazolo[3,2-a]pyrimidine derivatives of potential biological activities

In continuation to our previous work, thiazolopyrimidines 2a-x were synthesized through intramolecular cyclization of 2-phenacylthio-dihydropyrimidine hydrobromides 1a-x using polyphosphoric acid. On the other hand, thiazolo[3,2-a]pyrimidine-3-one 3 was coupled with aryldiazonium salts or condensed...

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Главные авторы:	Samia G. Abdel Moty (Автор), Mostafa A. Hussein (Автор), Salah A. Abdel Aziz (Автор), Mahrous A. Abou-Salim (Автор)
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Опубликовано:	Elsevier, 2016-03-01T00:00:00Z.
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