⁶⁸Ga-Radiolabeling and Pharmacological Characterization of a Kit-Based Formulation of the Gastrin-Releasing Peptide Receptor (GRP-R) Antagonist RM2 for Convenient Preparation of [⁶⁸Ga]Ga-RM2

• Главные авторы: Adrien Chastel (Автор), Delphine Vimont (Автор), Stephane Claverol (Автор), Marion Zerna (Автор), Sacha Bodin (Автор), Mathias Berndt (Автор), Stéphane Chaignepain (Автор), Elif Hindié (Автор), Clément Morgat (Автор)
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• Опубликовано: MDPI AG, 2021-07-01T00:00:00Z.
• Предметы: article
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Background: [⁶⁸Ga]Ga-RM2 is a potent Gastrin-Releasing Peptide-receptor (GRP-R) antagonist for imaging prostate cancer and breast cancer, currently under clinical evaluation in several specialized centers around the world. Targeted radionuclide therapy of GRP-R-expressing tumo...