<i>In Silico</i>-Motivated Discovery of Novel Potent Glycogen Synthase-3 Inhibitors: 1-(Alkyl/arylamino)-3H-naphtho[1,2,3-de]quinoline-2,7-dione Identified as a Scaffold for Kinase Inhibitor Development

Glycogen synthase kinase-3 (GSK-3) isoforms α and β have diverse roles within cell biology, and have been linked with multiple diseases that include prominent CNS conditions such as Alzheimer's disease and several psychiatric disorders. In this study, motivated by computation, we aimed to ident...

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Autores principales: Thomas D. Emmerich (Autor), Joseph M. Hayes (Autor)
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Publicado: MDPI AG, 2023-04-01T00:00:00Z.
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3rd Floor Main Library

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