Licraside as novel potent FXR agonist for relieving cholestasis: structure-based drug discovery and biological evaluation studies

Cholestasis is a common clinical disease caused by a disorder in bile acids (BAs) homeostasis, which promotes its development. The Farnesoid X receptor (FXR) plays a critical role in regulating BAs homeostasis, making it an essential target for cholestasis treatment. Although several active FXR agon...

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Main Authors: Lili Xi (Author), Axi Shi (Author), Tiantian Shen (Author), Guoxu Wang (Author), Yuhui Wei (Author), Jingjing Guo (Author)
Format: Book
Published: Frontiers Media S.A., 2023-06-01T00:00:00Z.
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3rd Floor Main Library

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