Recent Advances in Covalent Drug Discovery
In spite of the increasing number of biologics license applications, the development of covalent inhibitors is still a growing field within drug discovery. The successful approval of some covalent protein kinase inhibitors, such as ibrutinib (BTK covalent inhibitor) and dacomitinib (EGFR covalent in...
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MDPI AG,
2023-04-01T00:00:00Z.
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