Design and Microwave Synthesis of New (5<i>Z</i>) 5-Arylidene-2-thioxo-1,3-thiazolinidin-4-one and (5<i>Z</i>) 2-Amino-5-arylidene-1,3-thiazol-4(5<i>H</i>)-one as New Inhibitors of Protein Kinase DYRK1A

• 主要な著者: Khadidja Bourahla (著者), Solène Guihéneuf (著者), Emmanuelle Limanton (著者), Ludovic Paquin (著者), Rémy Le Guével (著者), Thierry Charlier (著者), Mustapha Rahmouni (著者), Emilie Durieu (著者), Olivier Lozach (著者), François Carreaux (著者), Laurent Meijer (著者), Jean-Pierre Bazureau (著者)
• フォーマット: 図書
• 出版事項: MDPI AG, 2021-10-01T00:00:00Z.
• 主題: article
• オンライン･アクセス: Connect to this object online.

Here, we report on the synthesis of libraries of new 5-arylidene-2-thioxo-1,3-thiazolidin-4-ones 3 (twenty-two compounds) and new 2-amino-5-arylidene-1,3-thiazol-4(5<i>H</i>)-ones 5 (twenty-four compounds) with stereo controlled <i>Z</i>-geometry under microwave irradiation....